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BRENDA support

Literature summary for 2.4.1.37 extracted from

  • Strecker, C.; Peters, H.; Hackl, T.; Peters, T.; Meyer, B.
    Fragment growing to design optimized inhibitors for human blood group B galactosyltransferase (GTB) (2019), ChemMedChem, 14, 1336-1342 .
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
1-(3-phenyl-1,2,4-thiadiazol-5-yl)piperazine
-
Homo sapiens
1-[3-(naphthalen-1-yl)-1,2,4-thiadiazol-5-yl]piperazine
-
Homo sapiens

Organism

Organism UniProt Comment Textmining
Homo sapiens P16442
-
-

Source Tissue

Source Tissue Comment Organism Textmining

Ki Value [mM]

Ki Value [mM] Ki Value maximum [mM] Inhibitor Comment Organism Structure
0.271
-
1-[3-(naphthalen-1-yl)-1,2,4-thiadiazol-5-yl]piperazine pH not specified in the publication, temperature not specified in the publication Homo sapiens
0.8
-
1-(3-phenyl-1,2,4-thiadiazol-5-yl)piperazine pH not specified in the publication, temperature not specified in the publication Homo sapiens