Inhibitors | Comment | Organism | Structure |
---|---|---|---|
additional information | no inhibition by N-[4-[5-(2,4-diamino-6-oxo-1,6-dihydropyrimidin-5-yl)-2-(2,2,2-trifluoroacetyl)pentyl]benzoyl]-L-glutamic acid | Escherichia coli | |
N-[4-[5-(2,4-diamino-6-oxo-1,6-dihydropyrimidin-5-yl)-2-(2,2,2-trifluoroacetyl)pentyl]benzoyl]-L-glutamic acid | effective inhibitor | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Escherichia coli | - |
- |
- |
Homo sapiens | - |
recombinant | - |
Synonyms | Comment | Organism |
---|---|---|
GAR TFase | - |
Escherichia coli |
GAR TFase | - |
Homo sapiens |
glycinamide ribonucleotide transformylase | - |
Escherichia coli |
glycinamide ribonucleotide transformylase | - |
Homo sapiens |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.0005 | - |
N-[4-[5-(2,4-diamino-6-oxo-1,6-dihydropyrimidin-5-yl)-2-(2,2,2-trifluoroacetyl)pentyl]benzoyl]-L-glutamic acid | 26°C, pH 7.5 | Homo sapiens |