Cloned (Comment) | Organism |
---|---|
human-derived gene is expressed in Escherichia coli | Pneumocystis carinii |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
methotrexate | - |
Pneumocystis carinii | |
pyrimethamine | poor inhibitor | Pneumocystis carinii | |
trimethoprim | poor inhibitor | Pneumocystis carinii | |
trimetrexate | - |
Pneumocystis carinii |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.0027 | - |
7,8-dihydrofolate | recombinant from E. coli | Pneumocystis carinii | |
0.0043 | - |
NADPH | recombinant from E. coli | Pneumocystis carinii |
Molecular Weight [Da] | Molecular Weight Maximum [Da] | Comment | Organism |
---|---|---|---|
25000 | - |
SDS-PAGE and DNA-sequence determination | Pneumocystis carinii |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Pneumocystis carinii | - |
human-derived | - |
Purification (Comment) | Organism |
---|---|
recombinant purified from Escherichia coli | Pneumocystis carinii |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.000000016 | - |
methotrexate | recombinant enzyme derived from E. coli | Pneumocystis carinii | |
0.00000023 | - |
trimetrexate | recombinant enzyme derived from E. coli | Pneumocystis carinii | |
0.000065 | - |
pyrimethamine | recombinant enzyme derived from E. coli | Pneumocystis carinii | |
0.00028 | - |
trimethoprim | recombinant enzyme derived from E. coli | Pneumocystis carinii |