Cloned (Comment) | Organism |
---|---|
expression in Sf9 cell | Homo sapiens |
Protein Variants | Comment | Organism |
---|---|---|
C132A | no catalytic activity, part of CXXC motif | Homo sapiens |
C135A | no catalytic activity, part of CXXC motif | Homo sapiens |
C16A | 40% of wild-type activity | Homo sapiens |
C43A | 35% of wild-type activity. C43 can form a disulfide bond with C51 | Homo sapiens |
C43A/C51A | 112% of wild-type activity | Homo sapiens |
C51A | 95% of wild-type activity. C43 can form a disulfide bond with C51 | Homo sapiens |
C85A | 100% of wild-type activity | Homo sapiens |
C96A | 45% of wild-type activity | Homo sapiens |
DELTAC43-C51 | 85% of wild-type activity | Homo sapiens |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
warfarin | - |
Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.004 | - |
warfarin | wild-type, pH 8.6, 30°C | Homo sapiens | |
0.012 | - |
warfarin | mutant C43A, pH 8.6, 30°C | Homo sapiens |