Ligand ketoconazole 2R,4R enantiomer
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Basic Ligand Information
C26H28ClN4O4
ketoconazole 2R,4R enantiomer
XMAYWYJOQHXEEK-BVAGGSTKSA-N
Roles as Enzyme Ligand
Inhibitor in Enzyme-catalyzed Reactions (1 result)
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Enzyme Kinetic Parameters
IC50 Value (1 result)
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References & Links
Literature References (1)
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Inhibition of CYP3A4 and CYP3A5 catalyzed metabolism of alprazolam and quinine by ketoconazole as racemate and four different enantiomers
2007
Allqvist, A.; Miura, J.; Bertilsson, L.; Mirghani, R.A.
Eur. J. Clin. Pharmacol.
63
173-179
Links to other databases for ketoconazole 2R,4R enantiomer