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Design, synthesis and evaluation of isaindigotone derivatives as acetylcholinesterase and butyrylcholinesterase inhibitors
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Acetylcholinesterase inhibitors from the toadstool Cortinarius infractus
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Tacrine-based dual binding site acetylcholinesterase inhibitors as potential disease-modifying anti-Alzheimer drug candidates
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Acetylcholinesterase inhibitory pyridine alkaloids of the leaves of Senna multijuga
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Synthesis and in vitro evaluation of N-alkyl-7-methoxytacrine hydrochlorides as potential cholinesterase inhibitors in Alzheimer disease
2010
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Probing the mid-gorge of cholinesterases with spacer-modified bivalent quinazolinimines leads to highly potent and selective butyrylcholinesterase inhibitors
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The characterization of Lucilia cuprina acetylcholinesterase as a drug target, and the identification of novel inhibitors by high throughput screening
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Crystal structures of human cholinesterases in complex with huprine W and tacrine: elements of specificity for anti-Alzheimers drugs targeting acetyl- and butyryl-cholinesterase
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Synthesis, biological activity and molecular modeling studies on 1H-benzimidazole derivatives as acetylcholinesterase inhibitors
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Allosteric inhibitors of the NS3 protease from the hepatitis C virus
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Inhibition of cholinesterase and monoamine oxidase-B activity by tacrine-homoisoflavonoid hybrids
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