Ligand N-[(furan-2-yl)methyl]-1-[(3S)-1,2,3,4-tetrahydroisoquinoline-3-carbonyl]piperidine-4-carboxamide
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Basic Ligand Information
C21H25N3O3
N-[(furan-2-yl)methyl]-1-[(3S)-1,2,3,4-tetrahydroisoquinoline-3-carbonyl]piperidine-4-carboxamide
CHWQZRDDUSGKFB-IBGZPJMESA-N
Roles as Enzyme Ligand
Inhibitor in Enzyme-catalyzed Reactions (1 result)
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SETDB1-TTD inhibitor, binds in the aromatic cage
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Enzyme Kinetic Parameters
References & Links
Literature References (1)
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SETDB1, an H3K9-specific methyltransferase An attractive epigenetic target to combat cancer
2024
Prashanth, S.; Radha Maniswami, R.; Rajajeyabalachandran, G.; Jegatheesan, S.K.
Drug Discov. Today
29
103982
Links to other databases for N-[(furan-2-yl)methyl]-1-[(3S)-1,2,3,4-tetrahydroisoquinoline-3-carbonyl]piperidine-4-carboxamide