Ligand 1-[(3,4-dimethoxyphenyl)methyl]-4-[[2-(trifluoromethyl)-7H-pyrrolo[2,3-b]pyridin-7-yl]methyl]piperidin-4-ol

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Basic Ligand Information

Molecular Structure

C₂₃H₂₆F₃N₃O₃

1-[(3,4-dimethoxyphenyl)methyl]-4-[[2-(trifluoromethyl)-7H-pyrrolo[2,3-b]pyridin-7-yl]methyl]piperidin-4-ol

YYLNGHCBPXQZBL-UHFFFAOYSA-N

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Roles as Enzyme Ligand

Inhibitor in Enzyme-catalyzed Reactions (1 result)

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2.1.1.366

peptidecompetitive SETDB1 inhibitor, decreases SETDB1/ESET levels without changing the mRNA levels (FRET) and exerts noticeable inhibitory effects on H3K9 trimethylation. Induces neuronal cytotoxicity at 0.1 mM

777166

Enzyme Kinetic Parameters

References & Links

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Show Reference (1 entry)

Links to other databases for 1-[(3,4-dimethoxyphenyl)methyl]-4-[[2-(trifluoromethyl)-7H-pyrrolo[2,3-b]pyridin-7-yl]methyl]piperidin-4-ol

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PubChem

UniChem