Ligand 1-methyl-5H-[1,2,4]triazolo[4,3-a][3,1]benzoxazine
Please wait a moment until all data is loaded. This message will disappear when all data is loaded.
Basic Ligand Information
C10H9N3O
1-methyl-5H-[1,2,4]triazolo[4,3-a][3,1]benzoxazine
YSNQHWRZFNUYIK-UHFFFAOYSA-N
Roles as Enzyme Ligand
Inhibitor in Enzyme-catalyzed Reactions (1 result)
Please wait a moment until the data is sorted. This message will disappear when the data is sorted.
SETDB1-TTD inhibitor, binds to the acetyl lysine (Kac) pocket of the SETDB1-TTD
-
Enzyme Kinetic Parameters
References & Links
Literature References (1)
Please wait a moment until the data is sorted. This message will disappear when the data is sorted.
SETDB1, an H3K9-specific methyltransferase An attractive epigenetic target to combat cancer
2024
Prashanth, S.; Radha Maniswami, R.; Rajajeyabalachandran, G.; Jegatheesan, S.K.
Drug Discov. Today
29
103982
Links to other databases for 1-methyl-5H-[1,2,4]triazolo[4,3-a][3,1]benzoxazine