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Ligand (4-chloro-3-(N,N-dimethylsulfamoyl)phenyl)methanesulfonyl fluoride

Basic Ligand Information

Molecular Structure

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Roles as Enzyme Ligand

Inhibitor in Enzyme-catalyzed Reactions (1 result)

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Show Inhibitors (1 entry)

EC NUMBER

COMMENTARY

LITERATURE

ENZYME 3D STRUCTURE

2.5.1.18

-

759613

-

Enzyme Kinetic Parameters

IC₅₀ Value (1 result)

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Show IC50 Value (1 entry)

EC NUMBER

IC50 VALUE

IC50 VALUE MAXIMUM

COMMENTARY

LITERATURE

2.5.1.18

0.0008

-

at pH 8.0 and 37°C

759613

References & Links

Literature References (1)

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Show Reference (1 entry)

BRENDA REFERENCE ID

PUBMED ID

TITLE

YEAR

AUTHORS

JOURNAL

VOLUME

PAGES

759613

32105470

Development of benzenesulfonamide derivatives as potent glutathione transferase omega-1 inhibitors

2020

Xie, Y.; Tummala, P.; Oakley, A.J.; Deora, G.S.; Nakano, Y.; Rooke, M.; Cuellar, M.E.; Strasser, J.M.; Dahlin, J.L.; Walters, M.A.; Casarotto, M.G.; Board, P.G.; Baell, J.B.

J. Med. Chem.

63

2894-2914

Links to other databases for (4-chloro-3-(N,N-dimethylsulfamoyl)phenyl)methanesulfonyl fluoride

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