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BRENDA support

Ligand K-252a

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Basic Ligand Information

Molecular Structure
Picture of K-252a (click for magnification)
Molecular Formula
BRENDA Name
InChIKey
C27H21N3O5
K-252a
KOZFSFOOLUUIGY-SOLYNIJKSA-N
Synonyms:
K252a
Pathway Source
Pathways

Roles as Enzyme Ligand

Inhibitor in Enzyme-catalyzed Reactions (9 results)

EC NUMBER
COMMENTARY
LITERATURE
ENZYME 3D STRUCTURE
complete inhibition at 200 nM
-
strong inhibition
-
inhibits CaM-KII
-
microbial broth product, highly selective
-
a potent inhibitor of protein kinase
-

3D Structure of Enzyme-Ligand-Complex (PDB) (8 results)

Enzyme Kinetic Parameters

IC50 Value (2 results)

EC NUMBER
IC50 VALUE
IC50 VALUE MAXIMUM
COMMENTARY
LITERATURE

References & Links

Links to other databases for K-252a

ChEBI
PubChem
ChEBI
PubChem