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ampicillin + H2O
(2R,4S)-2-[(R)-[[(2R)-2-amino-2-phenylacetyl]amino](carboxy)methyl]-5,5-dimethyl-1,3-thiazolidine-4-carboxylic acid
azlocillin + H2O
(2R,4S)-2-[(R)-carboxy({(2R)-2-[(2-oxoimidazolidine-1-carbonyl)amino]-2-phenylacetyl}amino)methyl]-5,5-dimethyl-1,3-thiazolidine-4-carboxylic acid
-
-
-
-
?
biapenem + H2O
(4R,5S)-5-[(1S,2R)-1-carboxy-2-hydroxypropyl]-3-[(6,7-dihydro-5H-pyrazolo[1,2-a][1,2,4]triazol-4-ium-6-yl)sulfanyl]-4-methyl-4,5-dihydro-1H-pyrrole-2-carboxylate
cefaclor + H2O
(2R)-2-[(R)-{[(2R)-2-amino-2-phenylacetyl]amino}(carboxy)methyl]-5-chloro-3,6-dihydro-2H-1,3-thiazine-4-carboxylic acid
cefadroxil + H2O
(2R)-2-[(R)-{[(2R)-2-amino-2-(4-hydroxyphenyl)acetyl]amino}(carboxy)methyl]-5-methyl-3,6-dihydro-2H-1,3-thiazine-4-carboxylic acid
-
-
-
-
?
cefazolin + H2O
(2R)-2-[(R)-carboxy[2-(1H-tetrazol-1-yl)acetamido]methyl]-5-[[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]methyl]-3,6-dihydro-2H-1,3-thiazine-4-carboxylic acid
-
-
-
?
cefepime + H2O
(2R)-2-[(R)-[[(2Z)-2-(2-amino-1,3-thiazol-4-yl)-2-(methoxyimino)acetyl]amino](carboxy)methyl]-5-[(1-methylpyrrolidinium-1-yl)methyl]-3,6-dihydro-2H-1,3-thiazine-4-carboxylate
-
-
-
-
?
cefmetazole + H2O
(2R)-2-[(S)-carboxy{2-[(cyanomethyl)sulfanyl]acetamido}methoxymethyl]-5-{[(1-methyl-1H-tetrazol-5-yl)sulfanyl]methyl}-3,6-dihydro-2H-1,3-thiazine-4-carboxylic acid
-
-
-
-
?
cefotaxime + H2O
(2R)-5-[(acetyloxy)methyl]-2-[(R)-[[(2E)-2-(2-amino-1,3-thiazol-4-yl)-2-(methoxyimino)acetyl]amino](carboxy)methyl]-3,6-dihydro-2H-1,3-thiazine-4-carboxylic acid
-
-
-
-
?
cefoxitin + H2O
(2R)-5-[(carbamoyloxy)methyl]-2-[(S)-carboxy(methoxy)[(thiophen-2-ylacetyl)amino]methyl]-3,6-dihydro-2H-1,3-thiazine-4-carboxylic acid
cefprozil + H2O
(2R)-2-[(R)-{[(2R)-2-amino-2-(4-hydroxyphenyl)acetyl]amino}(carboxy)methyl]-5-[(1E)-prop-1-en-1-yl]-3,6-dihydro-2H-1,3-thiazine-4-carboxylic acid
-
-
-
-
?
cefsulodin + H2O
(2R)-5-[(4-carbamoylpyridin-1-ium-1-yl)methyl]-2-[(R)-carboxy{[(2R)-2-phenyl-2-sulfoacetyl]amino}methyl]-3,6-dihydro-2H-1,3-thiazine-4-carboxylate
-
-
-
-
?
ceftizoxime + H2O
(2R)-2-[(R)-{[(2Z)-2-(2-amino-1,3-thiazol-4-yl)-2-(methoxyimino)acetyl]amino}(carboxy)methyl]-3,6-dihydro-2H-1,3-thiazine-4-carboxylic acid
-
-
-
-
?
cefuroxime + H2O
(2R)-5-[(carbamoyloxy)methyl]-2-[(R)-carboxy{[(2Z)-2-(furan-2-yl)-2-(methoxyimino)acetyl]amino}methyl]-3,6-dihydro-2H-1,3-thiazine-4-carboxylic acid
-
-
-
-
?
cephaloridine + H2O
(2R)-2-[(R)-carboxy[(thiophen-2-ylacetyl)amino]methyl]-5-(pyridinium-1-ylmethyl)-3,6-dihydro-2H-1,3-thiazine-4-carboxylate
-
-
-
-
?
cephalosporin C + H2O
N6-[(R)-{(2R)-5-[(acetyloxy)methyl]-4-carboxy-3,6-dihydro-2H-1,3-thiazin-2-yl}(carboxy)methyl]-6-oxo-D-lysine
-
-
-
-
?
cephalothin + H2O
(2R)-5-[(acetyloxy)methyl]-2-[(R)-carboxy[(thiophen-2-ylacetyl)amino]methyl]-3,6-dihydro-2H-1,3-thiazine-4-carboxylic acid
-
-
-
-
?
cephalotin + H2O
(2R)-5-[(acetyloxy)methyl]-2-[(R)-carboxy[(thiophen-2-ylacetyl)amino]methyl]-3,6-dihydro-2H-1,3-thiazine-4-carboxylic acid
-
-
-
?
cephradine + H2O
(2R)-2-[(R)-{[(2R)-2-amino-2-(cyclohexa-1,4-dien-1-yl)acetyl]amino}(carboxy)methyl]-5-methyl-3,6-dihydro-2H-1,3-thiazine-4-carboxylic acid
-
-
-
-
?
clavulanic acid + H2O
(2R,4R,5Z)-2-(carboxymethyl)-5-(2-hydroxyethylidene)-1,3-oxazolidine-4-carboxylic acid
-
-
-
-
?
imipenem + H2O
(5R)-5-[(1S,2R)-1-carboxy-2-hydroxypropyl]-3-([2-[(iminomethyl)amino]ethyl]sulfanyl)-4,5-dihydro-1H-pyrrole-2-carboxylic acid
-
-
-
?
imipenem + H2O
(5R)-5-[(1S,2R)-1-carboxy-2-hydroxypropyl]-3-({2-[(iminomethyl)amino]ethyl}sulfanyl)-4,5-dihydro-1H-pyrrole-2-carboxylic acid
-
-
-
?
meropenem + H2O
(4R,5S)-5-[(1S,2R)-1-carboxy-2-hydroxypropyl]-3-{[(3S,5S)-5-(dimethylcarbamoyl)pyrrolidin-3-yl]sulfanyl}-4-methyl-4,5-dihydro-1H-pyrrole-2-carboxylic acid
-
-
-
?
moxalactam + H2O
(2R)-2-{(R)-carboxy[2-carboxy(4-hydroxyphenyl)acetamido]methoxymethyl}-5-{[(1-methyl-1H-tetrazol-5-yl)sulfanyl]methyl}-3,6-dihydro-2H-1,3-oxazine-4-carboxylic acid
-
-
-
-
?
nitrocefin + H2O
(2R)-2-{(R)-carboxy[2-(thiophen-2-yl)acetamido]methyl}-5-[(E)-2-(2,4-dinitrophenyl)ethenyl]-3,6-dihydro-2H-1,3-thiazine-4-carboxylic acid
penicillin G + H2O
(2R,4S)-2-[(R)-carboxy[(phenylacetyl)amino]methyl]-5,5-dimethyl-1,3-thiazolidine-4-carboxylic acid
piperacillin + H2O
(2R,4S)-2-[(R)-carboxy[[(2R)-2-[[(4-ethyl-2,3-dioxopiperazin-1-yl)carbonyl]amino]-2-phenylacetyl]amino]methyl]-5,5-dimethyl-1,3-thiazolidine-4-carboxylic acid
-
-
-
-
?
ticarcillin + H2O
(2R,4S)-2-[(R)-carboxy[[(2R)-2-carboxy-2-(thiophen-3-yl)acetyl]amino]methyl]-5,5-dimethyl-1,3-thiazolidine-4-carboxylic acid
-
-
-
-
?
ampicillin + H2O
(2R,4S)-2-[(R)-[[(2R)-2-amino-2-phenylacetyl]amino](carboxy)methyl]-5,5-dimethyl-1,3-thiazolidine-4-carboxylic acid
-
-
-
-
?
ampicillin + H2O
(2R,4S)-2-[(R)-[[(2R)-2-amino-2-phenylacetyl]amino](carboxy)methyl]-5,5-dimethyl-1,3-thiazolidine-4-carboxylic acid
-
-
-
?
biapenem + H2O
(4R,5S)-5-[(1S,2R)-1-carboxy-2-hydroxypropyl]-3-[(6,7-dihydro-5H-pyrazolo[1,2-a][1,2,4]triazol-4-ium-6-yl)sulfanyl]-4-methyl-4,5-dihydro-1H-pyrrole-2-carboxylate
-
-
-
-
?
biapenem + H2O
(4R,5S)-5-[(1S,2R)-1-carboxy-2-hydroxypropyl]-3-[(6,7-dihydro-5H-pyrazolo[1,2-a][1,2,4]triazol-4-ium-6-yl)sulfanyl]-4-methyl-4,5-dihydro-1H-pyrrole-2-carboxylate
-
-
-
?
cefaclor + H2O
(2R)-2-[(R)-{[(2R)-2-amino-2-phenylacetyl]amino}(carboxy)methyl]-5-chloro-3,6-dihydro-2H-1,3-thiazine-4-carboxylic acid
-
-
-
-
?
cefaclor + H2O
(2R)-2-[(R)-{[(2R)-2-amino-2-phenylacetyl]amino}(carboxy)methyl]-5-chloro-3,6-dihydro-2H-1,3-thiazine-4-carboxylic acid
-
-
-
?
cefoxitin + H2O
(2R)-5-[(carbamoyloxy)methyl]-2-[(S)-carboxy(methoxy)[(thiophen-2-ylacetyl)amino]methyl]-3,6-dihydro-2H-1,3-thiazine-4-carboxylic acid
-
-
-
-
?
cefoxitin + H2O
(2R)-5-[(carbamoyloxy)methyl]-2-[(S)-carboxy(methoxy)[(thiophen-2-ylacetyl)amino]methyl]-3,6-dihydro-2H-1,3-thiazine-4-carboxylic acid
-
-
-
?
nitrocefin + H2O
(2R)-2-{(R)-carboxy[2-(thiophen-2-yl)acetamido]methyl}-5-[(E)-2-(2,4-dinitrophenyl)ethenyl]-3,6-dihydro-2H-1,3-thiazine-4-carboxylic acid
-
-
-
-
?
nitrocefin + H2O
(2R)-2-{(R)-carboxy[2-(thiophen-2-yl)acetamido]methyl}-5-[(E)-2-(2,4-dinitrophenyl)ethenyl]-3,6-dihydro-2H-1,3-thiazine-4-carboxylic acid
-
-
-
?
nitrocefin + H2O
(2R)-2-{(R)-carboxy[2-(thiophen-2-yl)acetamido]methyl}-5-[(E)-2-(2,4-dinitrophenyl)ethenyl]-3,6-dihydro-2H-1,3-thiazine-4-carboxylic acid
-
-
-
-
?
nitrocefin + H2O
(2R)-2-{(R)-carboxy[2-(thiophen-2-yl)acetamido]methyl}-5-[(E)-2-(2,4-dinitrophenyl)ethenyl]-3,6-dihydro-2H-1,3-thiazine-4-carboxylic acid
-
-
-
?
penicillin G + H2O
(2R,4S)-2-[(R)-carboxy[(phenylacetyl)amino]methyl]-5,5-dimethyl-1,3-thiazolidine-4-carboxylic acid
-
-
-
-
?
penicillin G + H2O
(2R,4S)-2-[(R)-carboxy[(phenylacetyl)amino]methyl]-5,5-dimethyl-1,3-thiazolidine-4-carboxylic acid
-
-
-
?
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1-(2S)-3-mercapto-2-methyl-propionyl-D-proline
competitive inhibitor
2,5-diphenyl-2H-pyrazol-3,4-dicarboxylic acid
-
2,5-diphenyl-3,4-furan dicarboxylic acid
-
2-(((3-mercapto-5-(2-methylphenyl)-4H-1,2,4-triazol-4-yl)imino)methyl)benzoic acid
most effective inhibitor
2-[[5-(2-hydroxyphenyl)-1,3,4-oxadiazol-2-yl]sulfanyl]-N-phenylacetamide
-
2-[[5-(2-hydroxyphenyl)-1,3,4-thiadiazol-2-yl]sulfanyl]-N-phenylacetamide
-
2-[[5-(2-hydroxyphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl]-N-phenylacetamide
-
bulgecin A
partial non-competitive inhibition
Cys-Val-His-Ser-Pro-Asn-Arg-Glu-Cys
-
mixed inhibition
galangin
-
flavonoid, inhibition is not reversible by addition of Zn2+, orientation in the active site, the 4-keto and the 5-hydroxy groups bind to the Zn1 atom of the enzyme
N-(1,3-benzothiazol-2-yl)-2-[[5-(2-hydroxyphenyl)-1,3,4-oxadiazol-2-yl]sulfanyl]acetamide
-
N-(1,3-benzothiazol-2-yl)-2-[[5-(2-hydroxyphenyl)-1,3,4-thiadiazol-2-yl]sulfanyl]acetamide
-
N-(1,3-benzothiazol-2-yl)-2-[[5-(2-hydroxyphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl]acetamide
-
N-(1,3-benzothiazol-2-yl)-2-[[5-(pyridin-3-yl)-1,3,4-oxadiazol-2-yl]sulfanyl]acetamide
-
N-(1,3-benzothiazol-2-yl)-2-[[5-(pyridin-3-yl)-1,3,4-thiadiazol-2-yl]sulfanyl]acetamide
-
N-(1,3-benzothiazol-2-yl)-2-[[5-(pyridin-3-yl)-4H-1,2,4-triazol-3-yl]sulfanyl]acetamide
-
N-(1,3-benzothiazol-2-yl)-2-[[5-(pyridin-4-yl)-1,3,4-oxadiazol-2-yl]sulfanyl]acetamide
-
N-(1,3-benzothiazol-2-yl)-2-[[5-(pyridin-4-yl)-1,3,4-thiadiazol-2-yl]sulfanyl]acetamide
-
N-(1,3-benzothiazol-2-yl)-2-[[5-(pyridin-4-yl)-4H-1,2,4-triazol-3-yl]sulfanyl]acetamide
-
N-phenyl-2-[[5-(pyridin-4-yl)-1,3,4-oxadiazol-2-yl]sulfanyl]acetamide
-
N-phenyl-2-[[5-(pyridin-4-yl)-1,3,4-thiadiazol-2-yl]sulfanyl]acetamide
-
N-phenyl-2-[[5-(pyridin-4-yl)-4H-1,2,4-triazol-3-yl]sulfanyl]acetamide
-
N-[(benzyloxy) carbonyl]-L-cysteinyl glycine
-
additional information
-
no inhibition: Cys-Val-His-Ser-Pro-Asn-Arg-Glu-Cys
-
additional information
development of eighteen diaryl-substituted azolylthioacetamides as New Delhi metallo-beta-lactamase-1 enzyme inhibitors, overview
-
additional information
-
development of eighteen diaryl-substituted azolylthioacetamides as New Delhi metallo-beta-lactamase-1 enzyme inhibitors, overview
-
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0.0089 - 0.15
cephalothin
0.022
clavulanic acid
-
-
0.0023 - 0.103
nitrocefin
0.038 - 0.384
penicillin G
0.055
ampicillin
wild-type enzyme, pH 7.0, 25°C
1.33
ampicillin
mutant D120N, pH 7.0, 25°C
0.032
biapenem
wild-type enzyme, pH 7.0, 25°C
0.045
biapenem
mutant D120C, pH 7.0, 25°C
0.081
biapenem
mutant D120S, pH 7.0, 25°C
0.128
biapenem
mutant D120N, pH 7.0, 25°C
0.013
cefaclor
wild-type enzyme, pH 7.0, 25°C
0.08
cefaclor
mutant D120S, pH 7.0, 25°C
0.098
cefaclor
mutant D120C, pH 7.0, 25°C
0.55
cefaclor
mutant D120N, pH 7.0, 25°C
0.0011
cefoxitin
wild-type enzyme, pH 7.0, 25°C
0.053
cefoxitin
mutant D120S, pH 7.0, 25°C
0.055
cefoxitin
mutant D120C, pH 7.0, 25°C
0.098
cefoxitin
mutant D120N, pH 7.0, 25°C
0.0089
cephalothin
wild-type enzyme, pH 7.0, 25°C
0.033
cephalothin
mutant D120C, pH 7.0, 25°C
0.046
cephalothin
mutant D120S, pH 7.0, 25°C
0.15
cephalothin
mutant D120N, pH 7.0, 25°C
0.057
Imipenem
wild-type enzyme, pH 7.0, 25°C
0.065
Imipenem
mutant D120C, pH 7.0, 25°C
0.094
Imipenem
mutant D120S, pH 7.0, 25°C
0.31
Imipenem
mutant D120N, pH 7.0, 25°C
0.015
meropenem
wild-type enzyme, pH 7.0, 25°C
0.06
meropenem
mutant D120C, pH 7.0, 25°C
0.07
meropenem
mutant D120N, pH 7.0, 25°C
0.097
meropenem
mutant D120S, pH 7.0, 25°C
0.0023
nitrocefin
lactamase ZnCo-L1, 1.0 Zn(2+), 1.0 Co(2+)
0.0036
nitrocefin
lactamase ZnFe-L1, 1.0 Zn(2+), 1.0 Fe(3+)
0.004
nitrocefin
lactamase ZnFe-L1, 1.2 Zn(2+), 0.9 Fe(3+)
0.004
nitrocefin
wild-typewith 1.90 equiv of Zn(2+)
0.0041
nitrocefin
wild-type enzyme, pH 7.0, 25°C
0.0043
nitrocefin
lactamase 1Co-L1, 0.9 Co(2+), 0.10 Zn(2+)
0.0055
nitrocefin
lactamase 1Zn-L1, 1.0 Zn(2+)
0.0059
nitrocefin
lactamase ZnZn-L1, 2.0 Zn(2+) added
0.015
nitrocefin
-
30°C, pH 8.0
0.018
nitrocefin
H116C, not applicable Zn(2+) content
0.02
nitrocefin
H116C with 0.85 equiv of Zn(2+)
0.02
nitrocefin
lactamase CoCo-L1, 1.80 Co(2+)
0.053
nitrocefin
lactamase 1Fe-L1, 0.9 Co(2+), 0.20 Zn(2+)
0.068
nitrocefin
mutant D120N, pH 7.0, 25°C
0.069
nitrocefin
mutant D120C, pH 7.0, 25°C
0.072
nitrocefin
H121C with 0.98 equiv of Zn(2+)
0.099
nitrocefin
H121C, not applicable Zn(2+) content
0.103
nitrocefin
mutant D120S, pH 7.0, 25°C
0.038
penicillin G
wild-type enzyme, pH 7.0, 25°C
0.384
penicillin G
mutant D120N, pH 7.0, 25°C
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0.01
ampicillin
below, mutant D120C, pH 7.0, 25°C
0.01
ampicillin
below, mutant D120S, pH 7.0, 25°C
77
ampicillin
mutant D120N, pH 7.0, 25°C
520
ampicillin
wild-type enzyme, pH 7.0, 25°C
0.3
biapenem
mutant D120C, pH 7.0, 25°C
0.5
biapenem
mutant D120S, pH 7.0, 25°C
3.6
biapenem
mutant D120N, pH 7.0, 25°C
134
biapenem
wild-type enzyme, pH 7.0, 25°C
0.28
cefaclor
mutant D120S, pH 7.0, 25°C
0.3
cefaclor
mutant D120C, pH 7.0, 25°C
6.3
cefaclor
mutant D120N, pH 7.0, 25°C
42
cefaclor
wild-type enzyme, pH 7.0, 25°C
0.34
cefoxitin
mutant D120S, pH 7.0, 25°C
0.56
cefoxitin
mutant D120C, pH 7.0, 25°C
1.53
cefoxitin
mutant D120N, pH 7.0, 25°C
1.9
cefoxitin
wild-type enzyme, pH 7.0, 25°C
0.31
cephalothin
mutant D120C, pH 7.0, 25°C
0.37
cephalothin
mutant D120S, pH 7.0, 25°C
8.1
cephalothin
mutant D120N, pH 7.0, 25°C
82
cephalothin
wild-type enzyme, pH 7.0, 25°C
0.36
Imipenem
mutant D120C, pH 7.0, 25°C
0.63
Imipenem
mutant D120S, pH 7.0, 25°C
15
Imipenem
mutant D120N, pH 7.0, 25°C
370
Imipenem
wild-type enzyme, pH 7.0, 25°C
0.29
meropenem
mutant D120C, pH 7.0, 25°C
0.75
meropenem
mutant D120S, pH 7.0, 25°C
10.6
meropenem
mutant D120N, pH 7.0, 25°C
157
meropenem
wild-type enzyme, pH 7.0, 25°C
0.028
nitrocefin
mutant D120S, pH 7.0, 25°C
0.18
nitrocefin
mutant D120C, pH 7.0, 25°C
2.54
nitrocefin
mutant D120N, pH 7.0, 25°C
2.6
nitrocefin
lactamase 1Fe-L1, 0.9 Co(2+), 0.20 Zn(2+)
11
nitrocefin
lactamase 1Co-L1, 0.9 Co(2+), 0.10 Zn(2+)
20
nitrocefin
lactamase ZnFe-L1, 1.0 Zn(2+), 1.0 Fe(3+)
24
nitrocefin
-
30°C, pH 8.0
24
nitrocefin
lactamase ZnFe-L1, 1.2 Zn(2+), 0.9 Fe(3+)
26
nitrocefin
lactamase ZnCo-L1, 1.0 Zn(2+), 1.0 Co(2+)
30
nitrocefin
lactamase 1Zn-L1, 1.0 Zn(2+)
39
nitrocefin
lactamase ZnZn-L1, 2.0 Zn(2+) added
41
nitrocefin
wild-type enzyme, pH 7.0, 25°C
63
nitrocefin
lactamase CoCo-L1, 1.80 Co(2+)
0.01
penicillin G
below, mutant D120C, pH 7.0, 25°C
0.01
penicillin G
below, mutant D120S, pH 7.0, 25°C
45
penicillin G
mutant D120N, pH 7.0, 25°C
600
penicillin G
wild-type enzyme, pH 7.0, 25°C
Please wait a moment until the data is sorted. This message will disappear when the data is sorted.
0.00034
2-[[5-(2-hydroxyphenyl)-1,3,4-oxadiazol-2-yl]sulfanyl]-N-phenylacetamide
pH and temperature not specified in the publication
0.00051
2-[[5-(2-hydroxyphenyl)-1,3,4-thiadiazol-2-yl]sulfanyl]-N-phenylacetamide
pH and temperature not specified in the publication
0.000073
2-[[5-(2-hydroxyphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl]-N-phenylacetamide
pH and temperature not specified in the publication
0.0025
bulgecin A
25°C, pH 7.0
0.009 - 0.016
Cys-Val-His-Ser-Pro-Asn-Arg-Glu-Cys
0.00065
N-(1,3-benzothiazol-2-yl)-2-[[5-(2-hydroxyphenyl)-1,3,4-oxadiazol-2-yl]sulfanyl]acetamide
pH and temperature not specified in the publication
0.0018
N-(1,3-benzothiazol-2-yl)-2-[[5-(2-hydroxyphenyl)-1,3,4-thiadiazol-2-yl]sulfanyl]acetamide
pH and temperature not specified in the publication
0.00025
N-(1,3-benzothiazol-2-yl)-2-[[5-(2-hydroxyphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl]acetamide
pH and temperature not specified in the publication
0.001
N-(1,3-benzothiazol-2-yl)-2-[[5-(pyridin-3-yl)-1,3,4-oxadiazol-2-yl]sulfanyl]acetamide
pH and temperature not specified in the publication
0.0014
N-(1,3-benzothiazol-2-yl)-2-[[5-(pyridin-3-yl)-1,3,4-thiadiazol-2-yl]sulfanyl]acetamide
pH and temperature not specified in the publication
0.00086
N-(1,3-benzothiazol-2-yl)-2-[[5-(pyridin-3-yl)-4H-1,2,4-triazol-3-yl]sulfanyl]acetamide
pH and temperature not specified in the publication
0.00082
N-(1,3-benzothiazol-2-yl)-2-[[5-(pyridin-4-yl)-1,3,4-oxadiazol-2-yl]sulfanyl]acetamide
pH and temperature not specified in the publication
0.00033
N-(1,3-benzothiazol-2-yl)-2-[[5-(pyridin-4-yl)-1,3,4-thiadiazol-2-yl]sulfanyl]acetamide
pH and temperature not specified in the publication
0.00034
N-(1,3-benzothiazol-2-yl)-2-[[5-(pyridin-4-yl)-4H-1,2,4-triazol-3-yl]sulfanyl]acetamide
pH and temperature not specified in the publication
0.00043 - 0.00051
N-phenyl-2-[[5-(pyridin-4-yl)-1,3,4-oxadiazol-2-yl]sulfanyl]acetamide
0.00038 - 0.00039
N-phenyl-2-[[5-(pyridin-4-yl)-1,3,4-thiadiazol-2-yl]sulfanyl]acetamide
0.00025 - 0.00054
N-phenyl-2-[[5-(pyridin-4-yl)-4H-1,2,4-triazol-3-yl]sulfanyl]acetamide
0.009
Cys-Val-His-Ser-Pro-Asn-Arg-Glu-Cys
-
30°C, pH 8.0, uncompetitive
0.016
Cys-Val-His-Ser-Pro-Asn-Arg-Glu-Cys
-
30°C, pH 8.0, competitive
0.00043
N-phenyl-2-[[5-(pyridin-4-yl)-1,3,4-oxadiazol-2-yl]sulfanyl]acetamide
pH and temperature not specified in the publication
0.00051
N-phenyl-2-[[5-(pyridin-4-yl)-1,3,4-oxadiazol-2-yl]sulfanyl]acetamide
pH and temperature not specified in the publication
0.00038
N-phenyl-2-[[5-(pyridin-4-yl)-1,3,4-thiadiazol-2-yl]sulfanyl]acetamide
pH and temperature not specified in the publication
0.00039
N-phenyl-2-[[5-(pyridin-4-yl)-1,3,4-thiadiazol-2-yl]sulfanyl]acetamide
pH and temperature not specified in the publication
0.00025
N-phenyl-2-[[5-(pyridin-4-yl)-4H-1,2,4-triazol-3-yl]sulfanyl]acetamide
pH and temperature not specified in the publication
0.00054
N-phenyl-2-[[5-(pyridin-4-yl)-4H-1,2,4-triazol-3-yl]sulfanyl]acetamide
pH and temperature not specified in the publication
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Crowder, M.W.; Walsh, T.R.; Banovic, L.; Pettit, M.; Spencer, J.
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2008
Stenotrophomonas maltophilia (P52700)
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Aeromonas veronii, Aeromonas veronii (O31272), Stenotrophomonas maltophilia (E9RIT0), Stenotrophomonas maltophilia, Bacteroides fragilis (P25910), Bacteroides fragilis
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