EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
|---|
   6.5.1.2 | 0.000007 |
- |
5,7-diamino-2-tert-butyl-4-[4-(hydroxymethyl)-1,3-thiazol-2-yl]-4a,8a-dihydropyrido[2,3-d]pyrimidine-6-carbonitrile |
at pH 7.4 and 20°C |
747273 |
| 6.5.1.2 | 0.00001 |
- |
2-(cyclopentyloxy)-3',5'-dideoxy-3'-[(3,5-dichlorophenyl)methyl]adenosine |
pH and temperature not specified in the publication |
747327 |
| 6.5.1.2 | 0.00001 |
- |
2-(cyclopentyloxy)-5'-deoxy-3'-O-(3,4-dichlorobenzyl)adenosine |
pH and temperature not specified in the publication |
727137 |
| 6.5.1.2 | 0.00001 |
- |
2-amino[1,4]benzodioxino[2,3-b]pyridine-3-carboxamide |
pH and temperature not specified in the publication |
749394 |
| 6.5.1.2 | 0.00001 |
- |
5'-deoxy-2-[(trans-4-methylcyclohexyl)oxy]adenosine |
pH and temperature not specified in the publication |
747327 |
| 6.5.1.2 | 0.00001 |
- |
5'-deoxy-5'-fluoro-2-[(trans-4-methylcyclohexyl)oxy]adenosine |
IC50 less 0.00001 mM, pH 7.5, 22°C |
713771 |
| 6.5.1.2 | 0.000013 |
- |
5,7-diamino-2-tert-butyl-4-(4H-1,2,3-triazol-4-yl)-4a,8a-dihydropyrido[2,3-d]pyrimidine-6-carbonitrile |
at pH 7.4 and 20°C |
747273 |
| 6.5.1.2 | 0.000015 |
- |
5,7-diamino-2-tert-butyl-4-cyclopentyl-4a,8a-dihydropyrido[2,3-d]pyrimidine-6-carbonitrile |
at pH 7.4 and 20°C |
747273 |
| 6.5.1.2 | 0.000019 |
- |
2-(cyclopentyloxy)-5'-deoxyadenosine |
pH 7.5, 22°C |
713771 |
| 6.5.1.2 | 0.000019 |
- |
4-([4-amino-2-[(2-methylcyclohexyl)oxy]-5-oxopyrido[2,3-d]pyrimidin-8(5H)-yl]methyl)benzoic acid |
pH and temperature not specified in the publication |
727142 |
