EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.4.21.1 | 0.00002 |
- |
PS-341 |
at 37°C for 1 h, in 20 mM Tris buffer, pH 8.0, 0.5 mM EDTA and 0.035% SDS |
707667 |
3.4.21.1 | 0.00007 |
- |
MG-132 |
at 37°C for 1 h, in 20 mM Tris buffer, pH 8.0, 0.5 mM EDTA and 0.035% SDS |
707667 |
3.4.21.1 | 0.00026 |
- |
cyanopeptolin 1027 |
pH 7.5, 37°C |
754584 |
3.4.21.1 | 0.00026 |
- |
cyanopeptolin 985 |
pH 7.5, 37°C |
754584 |
3.4.21.1 | 0.00028 |
- |
N-(tert-butoxycarbonyl)glycyl-N5-[(1R)-1-(dihydroxyboranyl)-3-methylbutyl]-N1-(naphthalen-2-ylmethyl)-L-glutamamide |
at 37°C for 1 h, in 20 mM Tris buffer, pH 8.0, 0.5 mM EDTA and 0.035% SDS |
707667 |
3.4.21.1 | 0.00038 |
- |
N-benzoyl-L-tyrosine ethyl ester |
- |
693716 |
3.4.21.1 | 0.00054 |
- |
N-(tert-butoxycarbonyl)glycyl-N1-benzyl-N5-[(1R)-1-(dihydroxyboranyl)-3-methylbutyl]-L-glutamamide |
at 37°C for 1 h, in 20 mM Tris buffer, pH 8.0, 0.5 mM EDTA and 0.035% SDS |
707667 |
3.4.21.1 | 0.00084 |
- |
N-(tert-butoxycarbonyl)-L-alanyl-N5-[(1R)-1-(dihydroxyboranyl)-3-methylbutyl]-N1-(naphthalen-2-ylmethyl)-L-glutamamide |
at 37°C for 1 h, in 20 mM Tris buffer, pH 8.0, 0.5 mM EDTA and 0.035% SDS |
707667 |
3.4.21.1 | 0.00147 |
- |
N-(tert-butoxycarbonyl)-L-phenylalanyl-N5-[(1R)-1-(dihydroxyboranyl)-3-methylbutyl]-N1-(naphthalen-2-ylmethyl)-L-glutamamide |
at 37°C for 1 h, in 20 mM Tris buffer, pH 8.0, 0.5 mM EDTA and 0.035% SDS |
707667 |
3.4.21.1 | 0.0015 |
- |
N-(tert-butoxycarbonyl)-L-leucyl-N5-[(1R)-1-(dihydroxyboranyl)-3-methylbutyl]-N1-(naphthalen-2-ylmethyl)-L-glutamamide |
at 37°C for 1 h, in 20 mM Tris buffer, pH 8.0, 0.5 mM EDTA and 0.035% SDS |
707667 |