EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
|---|
   2.7.11.17 | 0.0000333 |
- |
ARRKWQKTGHAVRAIGRLSS |
calmodulin antagonist peptide, IC50: 33.3 nM in H2O, 10.6 nM in buffer containing 0.1% w/v Tween 80 |
490801 |
| 2.7.11.17 | 0.02 |
- |
7H-benzimidazo(2,1-a)benz(de)isoquinoline-7-one-3-carboxylate |
30°C, pH 7.5, mutant enzyme P274E |
722711 |
| 2.7.11.17 | 0.039 |
- |
8-[(6-chloropyrimidin-4-yl)oxy]quinoline |
pH and temperature not specified in the publication, for HuH7 cells |
760861 |
| 2.7.11.17 | 0.04 |
- |
8-([6-[(5-methoxy-1H-benzimidazol-2-yl)sulfanyl]pyrimidin-4-yl]oxy)quinoline |
pH and temperature not specified in the publication, for HuH7 cells: 0.04 mM |
760861 |
| 2.7.11.17 | 0.046 |
- |
N-(4-methoxyphenyl)-6-(piperazin-1-yl)pyrimidin-4-amine |
HuH7 cells, Eagle's medium, pH not specified in the publication, 37°C |
740158 |
| 2.7.11.17 | 0.054 |
- |
7-([6-[(5-methoxy-1H-benzimidazol-2-yl)sulfanyl]pyrimidin-4-yl]oxy)-4-methyl-2H-1-benzopyran-2-one |
pH and temperature not specified in the publication, for HuH7 cells |
760861 |
| 2.7.11.17 | 0.055 |
- |
8-([6-[(naphthalen-2-yl)oxy]pyrimidin-4-yl]oxy)-1,4-dihydroquinoline |
pH and temperature not specified in the publication, for HuH7 cells |
760861 |
| 2.7.11.17 | 0.06 |
- |
6-[(5-methoxy-1H-benzimidazol-2-yl)sulfanyl]-N-(4-methoxyphenyl)pyrimidin-4-amine |
pH and temperature not specified in the publication, for HuH7 cells: 0.06 mM |
760861 |
| 2.7.11.17 | 0.072 |
- |
4-methyl-7-([6-[(quinolin-8-yl)oxy]pyrimidin-4-yl]oxy)-2H-1-benzopyran-2-one |
pH and temperature not specified in the publication, for HuH7 cells |
760861 |
| 2.7.11.17 | 0.104 |
- |
2-[4-[6-(quinolin-8-yloxy)pyrimidin-4-yl]piperazin-1-yl]benzonitrile |
HuH7 cells, Eagle's medium, pH not specified in the publication, 37°C |
740158 |
