EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
|---|
    1.14.19.1 | 0.00000004 |
- |
4-(ethylamino)-3-(2-hydroxyethoxy)-N-[5-[3-(trifluoromethyl)benzyl]-1,3-thiazol-2-yl]benzamide |
in 100 mM sodium phosphate, pH 7.4, at 37°C |
696685 |
| 1.14.19.1 | 0.00000004 |
- |
4-ethylamino-3-(2-hydroxyethoxy)-N-[5-(3-trifluoromethylbenzyl)thiazol-2-yl]benzamide |
in 250 mM sucrose, 150 mM KCl, 40 mM NaF, 5 mM MgCl2, 100 mM sodium phosphate, pH 7.4, at 37°C |
696685 |
| 1.14.19.1 | 0.00000005 |
- |
N-[2-[7-[[4-chloro-3-(trifluoromethyl)benzyl]amino]-3-(4-methoxyphenyl)-2-oxoquinoxalin-1(2H)-yl]ethyl]acetamide |
- |
696683 |
| 1.14.19.1 | 0.0000001 |
- |
N-(2-[7-[(3,4-dichlorobenzyl)amino]-3-(4-methoxyphenyl)-2-oxopyrido[3,4-b]pyrazin-1(2H)-yl]ethyl)acetamide |
- |
697825 |
| 1.14.19.1 | 0.0000001 |
- |
N-[5-(3,5-difluorobenzyl)-1,3-thiazol-2-yl]-3-(2-hydroxyethoxy)-4-methoxybenzamide |
in 100 mM sodium phosphate, pH 7.4, at 37°C |
696684 |
| 1.14.19.1 | 0.0000002 |
- |
N-[5-[4-fluoro-3-(trifluoromethyl)benzyl]-1,3-thiazol-2-yl]-3-(2-hydroxyethoxy)-4-methoxybenzamide |
in 100 mM sodium phosphate, pH 7.4, at 37°C |
696684 |
| 1.14.19.1 | 0.0000003 |
- |
N-[5-[3,5-bis(trifluoromethyl)benzyl]-1,3-thiazol-2-yl]-3-(2-hydroxyethoxy)-4-methoxybenzamide |
in 100 mM sodium phosphate, pH 7.4, at 37°C |
696685 |
| 1.14.19.1 | 0.0000004 |
- |
4-(ethylamino)-3-(2-hydroxyethoxy)-N-[5-[3-(trifluoromethyl)benzyl]-1,3-thiazol-2-yl]benzamide |
in 100 mM sodium phosphate, pH 7.4, at 37°C |
696685 |
| 1.14.19.1 | 0.0000004 |
- |
4-ethylamino-3-(2-hydroxyethoxy)-N-[5-(3-trifluoromethylbenzyl)thiazol-2-yl]benzamide |
in 250 mM sucrose, 150 mM KCl, 40 mM NaF, 5 mM MgCl2, 100 mM sodium phosphate, pH 7.4, at 37°C |
696685 |
| 1.14.19.1 | 0.0000005 |
- |
N-(2-[6-[(3,4-dichlorobenzyl)amino]-3-oxo-2,3-dihydro-4H-1,4-benzoxazin-4-yl]ethyl)-2-hydroxyacetamide |
- |
696683 |
