EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
5.6.1.3 | 0.000001 |
- |
N-(3-aminopropyl)-N-[(1R)-1-(3-benzyl-7-chloro-4-oxo-3,4-dihydroquinazolin-2-yl)-2-methylpropyl]-3-fluoro-4-methylbenzamide |
wild-type |
688256 |
5.6.1.3 | 0.0000017 |
- |
6-[4-(trifluoromethyl)phenyl]-3,4-dihydroquinolin-2(1H)-one |
wild-type, pH 6.8 |
689127 |
5.6.1.3 | 0.0000035 |
- |
N-[3-fluoro-4'-(trifluoromethyl)biphenyl-4-yl]sulfuric diamide |
wild-type |
688256 |
5.6.1.3 | 0.000006 |
- |
N-[3-fluoro-4'-(trifluoromethyl)biphenyl-4-yl]sulfuric diamide |
mutant D130V |
688256 |
5.6.1.3 | 0.0000062 |
- |
N-[4'-(trifluoromethyl)biphenyl-4-yl]sulfuric diamide |
wild-type |
688256 |
5.6.1.3 | 0.000007 |
- |
N-[4'-(trifluoromethyl)biphenyl-4-yl]sulfuric diamide |
mutant D130V |
688256 |
5.6.1.3 | 0.000066 |
- |
6-[4-(trifluoromethyl)phenyl]-3,4-dihydroquinolin-2(1H)-one |
mutant I299F, pH 6.8 |
689127 |
5.6.1.3 | 0.000109 |
- |
6-[4-(trifluoromethyl)phenyl]-3,4-dihydroquinolin-2(1H)-one |
mutant A356T, pH 6.8 |
689127 |
5.6.1.3 | 0.00011 |
- |
N-[4'-(trifluoromethyl)biphenyl-4-yl]methanesulfonamide |
mutant D130V |
688256 |
5.6.1.3 | 0.00012 |
- |
N-[4'-(trifluoromethyl)biphenyl-4-yl]methanesulfonamide |
wild-type |
688256 |