EC Number   |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
|---|
    2.4.2.8 | -999 |
- |
more |
kinetics for product inhibition in forward and reverse reaction, wild-type enzyme |
638415 |
| 2.4.2.8 | -999 |
- |
more |
kinetics of product inhibition in forward reaction |
638410 |
| 2.4.2.8 | -999 |
- |
more |
overview, inhibition constants for diverse purine nucleotides and analogues |
638400 |
| 2.4.2.8 | 0.00000065 |
- |
[(3S)-4-hydroxy-3-[([4-hydroxy-5H-pyrrolo[3,2-d]pyrimidin-7-yl]methyl)amino]butyl]phosphonic acid |
at pH 7.6 and 37°C |
735767 |
| 2.4.2.8 | 0.00000065 |
- |
[(3S)-4-hydroxy-3-[[(4-oxo-4,5-dihydro-3H-pyrrolo[3,2-d]pyrimidin-7-yl)methyl]amino]butyl]phosphonic acid |
pH 7.6, 37°C |
722020 |
| 2.4.2.8 | 0.0000012 |
- |
[(3R)-4-hydroxy-3-[([4-hydroxy-5H-pyrrolo[3,2-d]pyrimidin-7-yl]methyl)amino]butyl]phosphonic acid |
at pH 7.6 and 37°C |
735767 |
| 2.4.2.8 | 0.0000013 |
- |
[(1S)-1-hydroxy-2-[[(3R,4R)-4-(6-oxo-1,6-dihydro-9H-purin-9-yl)-1-(phosphonoacetyl)pyrrolidin-3-yl]oxy]ethyl]phosphonic acid |
pH not specified in the publication, 37°C |
758563 |
| 2.4.2.8 | 0.000002 |
- |
[(1S)-1-hydroxy-2-[[(3R,4R)-4-(6-oxo-1,6-dihydro-9H-purin-9-yl)-1-(phosphonoacetyl)pyrrolidin-3-yl]oxy]ethyl]phosphonic acid |
pH not specified in the publication, 37°C |
758563 |
| 2.4.2.8 | 0.0000024 |
- |
[(2R)-3-hydroxy-2-[([4-hydroxy-5H-pyrrolo[3,2-d]pyrimidin-7-yl]methyl)amino]propoxy]phosphonic acid |
at pH 7.6 and 37°C |
735767 |
| 2.4.2.8 | 0.000003 |
- |
[3R,4R]-4-guanin-9-yl-3-((S)-2-hydroxy-2-phosphonoethyl)oxy-1-N-(phosphonopropionyl)pyrrolidine |
pH not specified in the publication, 37°C |
758563 |
