EC Number |
BRENDA No. |
Title |
Journal |
Volume |
Pages |
Year |
Organism |
PubMed ID |
---|
3.4.21.106 | 753876 |
Alpha-methylacyl-CoA racemase and hepsin as urinary prostate cancer markers |
Int. J. Biol. Markers |
30 |
e401-e406 |
2015 |
Homo sapiens |
25982684 |
3.4.21.106 | 752938 |
Design and synthesis of dye-conjugated hepsin inhibitors |
Bioorg. Chem. |
89 |
102990 |
2019 |
Homo sapiens |
31136899 |
3.4.21.106 | 753485 |
Design, synthesis and biological evaluation of PSMA/hepsin-targeted heterobivalent ligands |
Eur. J. Med. Chem. |
118 |
208-218 |
2016 |
Homo sapiens |
27128184 |
3.4.21.106 | 754402 |
Discovery of selective matriptase and hepsin serine protease inhibitors useful chemical tools for cancer cell biology |
J. Med. Chem. |
62 |
480-490 |
2019 |
Homo sapiens |
30571119 |
3.4.21.106 | 752764 |
SERPINB12 is a slow-binding inhibitor of granzyme A and hepsin |
Biochemistry |
54 |
6756-6759 |
2015 |
Homo sapiens |
26497600 |
3.4.21.106 | 752986 |
Structure-based design, synthesis, and biological evaluation of Leu-Arg dipeptide analogs as novel hepsin inhibitors |
Bioorg. Med. Chem. Lett. |
26 |
310-314 |
2016 |
Homo sapiens |
26711145 |
3.4.21.106 | 752945 |
Structure-based discovery of small molecule hepsin and HGFA protease inhibitors Evaluation of potency and selectivity derived from distinct binding pockets |
Bioorg. Med. Chem. |
23 |
2328-2343 |
2015 |
Homo sapiens |
25882520 |
3.4.21.106 | 752981 |
Structure-guided discovery of 2-aryl/pyridin-2-yl-1H-indole derivatives as potent and selective hepsin inhibitors |
Bioorg. Med. Chem. Lett. |
25 |
5309-5314 |
2015 |
Homo sapiens |
26421993 |
3.4.21.106 | 753410 |
The serine protease hepsin mediates urinary secretion and polymerisation of Zona Pellucida domain protein uromodulin |
eLife |
4 |
e08887 |
2015 |
Mus musculus |
26673890 |
3.4.21.106 | 755460 |
The serine proteinase hepsin is an activator of pro-matrix metalloproteinases molecular mechanisms and implications for extracellular matrix turnover |
Sci. Rep. |
7 |
16693 |
2017 |
Homo sapiens |
29196708 |