EC Number |
BRENDA No. |
Title |
Journal |
Volume |
Pages |
Year |
Organism |
PubMed ID |
---|
2.7.11.15 | 760330 |
A high-affinity peptide substrate for G protein-coupled receptor kinase 2 (GRK2) |
Amino Acids |
51 |
973-976 |
2019 |
Homo sapiens |
31004228 |
2.7.11.15 | 760331 |
Design of substrates and inhibitors of G protein-coupled receptor kinase 2 (GRK2) based on its phosphorylation reaction |
Amino Acids |
52 |
863-870 |
2020 |
Homo sapiens |
32577910 |
2.7.11.15 | 760459 |
G protein-coupled receptor kinase 2 inhibition improves erectile function through amelioration of endothelial dysfunction and oxidative stress in a rat model of type 2 diabetes |
Asian J. Androl. |
21 |
74-79 |
2019 |
Rattus norvegicus |
30226217 |
2.7.11.15 | 760708 |
Hit-to-lead optimization and discovery of a potent, and orally bioavailable G protein coupled receptor kinase 2 (GRK2) inhibitor |
Bioorg. Med. Chem. Lett. |
30 |
127602 |
2020 |
Homo sapiens |
33038544 |
2.7.11.15 | 760474 |
Inhibitory effects of two G protein-coupled receptor kinases on the cell surface expression and signaling of the human adrenomedullin receptor |
Biochem. Biophys. Res. Commun. |
470 |
894-899 |
2016 |
Homo sapiens |
26820533 |
2.7.11.15 | 760897 |
Multistep virtual screening for rapid identification of G protein-coupled receptors kinase 2 inhibitors for heart failure treatment |
Chemometr. Intell. Lab. Syst. |
185 |
32-40 |
2019 |
Homo sapiens |
- |
2.7.11.15 | 662131 |
A G protein-coupled receptor kinase induces Xenopus oocyte maturation |
J. Biol. Chem. |
278 |
15809-15814 |
2003 |
Rattus norvegicus |
12600992 |
2.7.11.15 | 645024 |
Activation of beta-adrenergic receptor kinase during myocardial ischemia |
Circ. Res. |
79 |
455-460 |
1996 |
Rattus norvegicus |
8781479 |
2.7.11.15 | 703084 |
Adenoviral beta-adrenergic receptor kinase inhibitor gene transfer improves exercise capacity, cardiac contractility, and systemic inflammation in a model of pressure overload hypertrophy |
Cardiovasc. Drugs Ther. |
22 |
373-381 |
2008 |
Rattus norvegicus |
18690529 |
2.7.11.15 | 661500 |
Adenovirus-mediated expression of beta-adrenergic receptor kinase C-terminus reduces intimal hyperplasia and luminal stenosis of arteriovenous polytetrafluoroethylene grafts in pigs |
Circulation |
111 |
1679-1684 |
2005 |
Bos taurus |
15781730 |