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Literature summary extracted from

  • Homan, K.T.; Waldschmidt, H.V.; Glukhova, A.; Cannavo, A.; Song, J.; Cheung, J.Y.; Koch, W.J.; Larsen, S.D.; Tesmer, J.J.
    Crystal structure of G protein-coupled receptor kinase 5 in complex with a rationally designed inhibitor (2015), J. Biol. Chem., 290, 20649-20659.
    View publication on PubMedView publication on EuropePMC

Crystallization (Commentary)

EC Number Crystallization (Comment) Organism
2.7.11.16 in complex with CCG215022, hanging drop vapor diffusion method, using 100 mM HEPES, pH 7.5, 4% (v/v) ethylene glycol, and 12% (w/v) PEG3350 Bos taurus

Inhibitors

EC Number Inhibitors Comment Organism Structure
2.7.11.16 balanol
-
Bos taurus
2.7.11.16 CCG215022
-
Bos taurus
2.7.11.16 GSK180736A
-
Bos taurus
2.7.11.16 paroxetine
-
Bos taurus
2.7.11.16 Takeda103A
-
Bos taurus

Localization

EC Number Localization Comment Organism GeneOntology No. Textmining
2.7.11.16 nucleus
-
Bos taurus 5634
-

Natural Substrates/ Products (Substrates)

EC Number Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
2.7.11.16 ATP + [G-protein-coupled receptor] Bos taurus
-
ADP + [G-protein-coupled receptor]phosphate
-
?

Organism

EC Number Organism UniProt Comment Textmining
2.7.11.16 Bos taurus P43249
-
-

Purification (Commentary)

EC Number Purification (Comment) Organism
2.7.11.16 Ni-NTA column chromatography and S200 gel filtration Bos taurus

Source Tissue

EC Number Source Tissue Comment Organism Textmining
2.7.11.16 cardiomyocyte
-
Bos taurus
-

Substrates and Products (Substrate)

EC Number Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
2.7.11.16 ATP + [G-protein-coupled receptor]
-
Bos taurus ADP + [G-protein-coupled receptor]phosphate
-
?

Synonyms

EC Number Synonyms Comment Organism
2.7.11.16 G protein-coupled receptor kinase 5
-
Bos taurus
2.7.11.16 GRK5
-
Bos taurus