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Literature summary extracted from

  • Ahmed, M.; Batista, J.; Rocha, T.; Mazzanti, C.M.; Hassan, W.; Morsch, V.M.; Loro, V.L.; Thome, G.; Schetinger, M.R.
    Comparative study of the inhibitory effect of antidepressants on cholinesterase activity in Bungarus sindanus (krait) venom, human serum and rat striatum (2008), J. Enzyme Inhib. Med. Chem., 23, 912-917.
    View publication on PubMed

Inhibitors

EC Number Inhibitors Comment Organism Structure
3.1.1.8 clomipramine competitive inhibition Homo sapiens
3.1.1.8 ethopropazine specific inhibitor Homo sapiens
3.1.1.8 imipramine competitive inhibition Homo sapiens
3.1.1.8 paroxetine mixed-type inhibition Homo sapiens
3.1.1.8 sertraline mixed-type inhibition Homo sapiens

Localization

EC Number Localization Comment Organism GeneOntology No. Textmining
3.1.1.8 extracellular
-
Homo sapiens
-
-

Organism

EC Number Organism UniProt Comment Textmining
3.1.1.8 Homo sapiens
-
-
-

Source Tissue

EC Number Source Tissue Comment Organism Textmining
3.1.1.8 heart
-
Homo sapiens
-
3.1.1.8 intestine
-
Homo sapiens
-
3.1.1.8 kidney
-
Homo sapiens
-
3.1.1.8 liver
-
Homo sapiens
-
3.1.1.8 lung
-
Homo sapiens
-
3.1.1.8 serum
-
Homo sapiens
-

Substrates and Products (Substrate)

EC Number Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
3.1.1.8 acetylthiocholine + H2O detection with 5,5-dithiobis(2-nitrobenzoic acid) Homo sapiens ?
-
?

Synonyms

EC Number Synonyms Comment Organism
3.1.1.8 acyl choline acylhydrolase
-
Homo sapiens
3.1.1.8 BuChE
-
Homo sapiens
3.1.1.8 butyrylcholinesterase
-
Homo sapiens
3.1.1.8 non specific cholinesterase
-
Homo sapiens
3.1.1.8 pseudo cholinesterase
-
Homo sapiens

Temperature Optimum [°C]

EC Number Temperature Optimum [°C] Temperature Optimum Maximum [°C] Comment Organism
3.1.1.8 25
-
assay at Homo sapiens

pH Optimum

EC Number pH Optimum Minimum pH Optimum Maximum Comment Organism
3.1.1.8 7.5
-
assay at Homo sapiens