Cloned (Comment) | Organism |
---|---|
CA I and CA II cDNA expressed in Escherichia coli BL21 (DE3) | Homo sapiens |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
5-(2-chlorophenyl)-1,3,4-thiadiazole-2-sulfonamide | - |
Bos taurus | |
5-(2-chlorophenyl)-1,3,4-thiadiazole-2-sulfonamide | - |
Homo sapiens | |
acetazolamide | - |
Bos taurus | |
acetazolamide | - |
Homo sapiens | |
benzolamide | - |
Bos taurus | |
benzolamide | - |
Homo sapiens | |
chlorazolamide | - |
Bos taurus | |
chlorazolamide | - |
Homo sapiens | |
dorzolamide | - |
Bos taurus | |
dorzolamide | - |
Homo sapiens | |
ethoxzolamide | - |
Bos taurus | |
ethoxzolamide | - |
Homo sapiens | |
methazolamide | - |
Bos taurus | |
methazolamide | - |
Homo sapiens |
Localization | Comment | Organism | GeneOntology No. | Textmining |
---|---|---|---|---|
microsome | - |
Bos taurus | - |
- |
Metals/Ions | Comment | Organism | Structure |
---|---|---|---|
Zn2+ | - |
Homo sapiens | |
Zn2+ | - |
Bos taurus |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
H2CO3 | Homo sapiens | - |
CO2 + H2O | - |
r | |
H2CO3 | Bos taurus | - |
CO2 + H2O | - |
r |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Bos taurus | - |
- |
- |
Homo sapiens | - |
- |
- |
Purification (Comment) | Organism |
---|---|
- |
Homo sapiens |
- |
Bos taurus |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
lung | - |
Bos taurus | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
H2CO3 | - |
Homo sapiens | CO2 + H2O | - |
r | |
H2CO3 | - |
Bos taurus | CO2 + H2O | - |
r |
Synonyms | Comment | Organism |
---|---|---|
bCA IV | - |
Homo sapiens |
bCA IV | - |
Bos taurus |
CA | - |
Homo sapiens |
CA | - |
Bos taurus |
CA I | - |
Homo sapiens |
CA II | - |
Homo sapiens |
CA IV | - |
Homo sapiens |
carbonic anhydrase | - |
Homo sapiens |
carbonic anhydrase | - |
Bos taurus |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.000003 | - |
chlorazolamide | pH 7.4, 25°C, hCA II | Homo sapiens | |
0.000008 | - |
ethoxzolamide | pH 7.4, 25°C, hCA II | Homo sapiens | |
0.000009 | - |
dorzolamide | pH 7.4, 25°C, hCA II | Homo sapiens | |
0.000009 | - |
benzolamide | pH 7.4, 25°C, hCA II | Homo sapiens | |
0.000012 | - |
benzolamide | pH 7.4, 25°C, bCA IV | Bos taurus | |
0.000012 | - |
acetazolamide | pH 7.4, 25°C, hCA II | Homo sapiens | |
0.000013 | - |
ethoxzolamide | pH 7.4, 25°C, bCA IV | Bos taurus | |
0.000014 | - |
methazolamide | pH 7.4, 25°C, hCA II | Homo sapiens | |
0.000015 | - |
chlorazolamide | pH 7.4, 25°C, bCA IV | Bos taurus | |
0.000015 | - |
chlorazolamide | pH 7.4, 25°C, hCA I | Homo sapiens | |
0.000018 | - |
benzolamide | pH 7.4, 25°C, hCA I | Homo sapiens | |
0.000025 | - |
ethoxzolamide | pH 7.4, 25°C, hCA I | Homo sapiens | |
0.000043 | - |
dorzolamide | pH 7.4, 25°C, bCA IV | Bos taurus | |
0.00022 | - |
acetazolamide | pH 7.4, 25°C, bCA IV | Bos taurus | |
0.00024 | - |
methazolamide | pH 7.4, 25°C, bCA IV | Bos taurus | |
0.00078 | - |
methazolamide | pH 7.4, 25°C, hCA I | Homo sapiens | |
0.0009 | - |
acetazolamide | pH 7.4, 25°C, hCA I | Homo sapiens | |
0.05 | - |
dorzolamide | pH 7.4, 25°C, hCA I | Homo sapiens |