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Literature summary for 3.6.5.6 extracted from

  • Gupta, K.; Panda, D.
    Perturbation of microtubule polymerization by quercetin through tubulin binding: a novel mechanism of its antiproliferative activity (2002), Biochemistry, 41, 13029-13038.
    View publication on PubMed

Activating Compound

Activating Compound Comment Organism Structure
quercetin 0.05 mM, stimulates GTPase activity about 8fold, but inhibits polymerization of microtubules and specifically inhibits colchicine binding to tubulin Capra hircus

Organism

Organism UniProt Comment Textmining
Capra hircus
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