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Literature summary for 3.5.2.3 extracted from

  • Krungkrai, J.; Krungkrai, S.R.; Phakanont, K.
    Antimalarial activity of orotate analogs that inhibit dihydroorotase and dihydroorotate dehydrogenase (1992), Biochem. Pharmacol., 43, 1295-1301.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
5-aminoorotate
-
Plasmodium berghei
5-bromoorotate
-
Plasmodium berghei
5-Fluoroorotate
-
Plasmodium berghei
5-iodoorotate
-
Plasmodium berghei
5-Methylorotate
-
Plasmodium berghei
Orotate
-
Plasmodium berghei

KM Value [mM]

KM Value [mM] KM Value Maximum [mM] Substrate Comment Organism Structure
0.008
-
L-dihydroorotate
-
Plasmodium berghei

Organism

Organism UniProt Comment Textmining
Plasmodium berghei
-
-
-

Purification (Commentary)

Purification (Comment) Organism
-
Plasmodium berghei