Inhibitors | Comment | Organism | Structure |
---|---|---|---|
hydroxamate matrix metalloproteinase inhibitors | - |
Homo sapiens | |
MAG-181 | mercaptosulfide matrix metalloproteinase inhibitor | Homo sapiens | |
MAG-182 | mercaptosulfide matrix metalloproteinase inhibitor | Homo sapiens | |
matrix metalloproteinase inhibitor GM6001 | - |
Homo sapiens | |
YHJ-294-1 | mercaptosulfide matrix metalloproteinase inhibitor | Homo sapiens | |
YHJ-294-2 | mercaptosulfide matrix metalloproteinase inhibitor | Homo sapiens | |
YHJ-72 | mercaptosulfide matrix metalloproteinase inhibitor | Homo sapiens | |
YHJ-73 | mercaptosulfide matrix metalloproteinase inhibitor | Homo sapiens | |
YHJ-74 | mercaptosulfide matrix metalloproteinase inhibitor | Homo sapiens | |
YHJ-75 | mercaptosulfide matrix metalloproteinase inhibitor | Homo sapiens |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
proteins + H2O | Homo sapiens | - |
peptides | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Reaction | Comment | Organism | Reaction ID |
---|---|---|---|
proteolytic degradation of proteins | active site structure | Homo sapiens |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
proteins + H2O | - |
Homo sapiens | peptides | - |
? |
Synonyms | Comment | Organism |
---|---|---|
endometase | - |
Homo sapiens |
endometase/matrilysin-2 | - |
Homo sapiens |
M10.029 | Merops-ID | Homo sapiens |
matrix metalloproteinase-26 | - |
Homo sapiens |
MMP-26 | - |
Homo sapiens |
MMP-26/endometase/matrilysin-2 | - |
Homo sapiens |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
additional information | - |
additional information | - |
Homo sapiens | |
0.0000028 | - |
YHJ-294-2 | pH 7.5, 25°C | Homo sapiens | |
0.0000086 | - |
YHJ-75 | pH 7.5, 25°C | Homo sapiens | |
0.000017 | - |
MAG-182 | pH 7.5, 25°C | Homo sapiens | |
0.000028 | - |
YHJ-73 | pH 7.5, 25°C | Homo sapiens | |
0.000081 | - |
MAG-181 | pH 7.5, 25°C | Homo sapiens | |
0.000082 | - |
YHJ-74 | pH 7.5, 25°C | Homo sapiens | |
0.00016 | - |
YHJ-72 | pH 7.5, 25°C | Homo sapiens | |
0.00045 | - |
YHJ-294-1 | pH 7.5, 25°C | Homo sapiens |