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Literature summary for 3.4.24.86 extracted from

  • Souza, D.G.; Ferreira, F.L.; Fagundes, C.T.; Amaral, F.A.; Vieira, A.T.; Lisboa, R.A.; Andrade, M.V.; Trifilieff, A.; Teixeira, M.M.
    Effects of PKF242-484 and PKF241-466, novel dual inhibitors of TNF-alpha converting enzyme and matrix metalloproteinases, in a model of intestinal reperfusion injury in mice (2007), Eur. J. Pharmacol., 571, 72-80.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
additional information not inhibited by FN-439 Mus musculus
PKF241-466 maximum inhibition at 10 mg/kg Mus musculus
PKF242-484 maximum inhibition at 10 mg/kg Mus musculus

Organism

Organism UniProt Comment Textmining
Mus musculus
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
p75 tumour necrosis factor receptor + H2O
-
Mus musculus ?
-
?
proTNF-alpha + H2O
-
Mus musculus soluble TNF-alpha
-
?

Synonyms

Synonyms Comment Organism
TACE
-
Mus musculus
TNF-alpha converting enzyme
-
Mus musculus