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Literature summary for 3.4.24.82 extracted from

  • Mosyak, L.; Georgiadis, K.; Shane, T.; Svenson, K.; Hebert, T.; McDonagh, T.; Mackie, S.; Olland, S.; Lin, L.; Zhong, X.; Kriz, R.; Reifenberg, E.L.; Collins-Racie, L.A.; Corcoran, C.; Freeman, B.; Zollner, R.; Marvell, T.; Vera, M.; Sum, P.E.; Lavallie, E.R.; Stahl, M.; Somers, W.
    Crystal structures of the two major aggrecan degrading enzymes, ADAMTS4 and ADAMTS5 (2008), Protein Sci., 17, 16-21.
    View publication on PubMedView publication on EuropePMC

Cloned(Commentary)

Cloned (Comment) Organism
expressed in CHO cells Homo sapiens

Crystallization (Commentary)

Crystallization (Comment) Organism
vapour diffusion method with 10% PEG 4K, 0.1 M MES (pH 6.0) Homo sapiens

Inhibitors

Inhibitors Comment Organism Structure
batimastat
-
Homo sapiens

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-

Purification (Commentary)

Purification (Comment) Organism
polypropyl aspartamide hydrophobic interaction column chromatography, gel filtration, anti-Flag M2 affinity chromatogaphy, and Mono Q column chromatography Homo sapiens

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
Abz-TEGEARGSVI-Dap(2,4-dinitrophenyl)-KK + H2O
-
Homo sapiens ?
-
?
aggrecan + H2O
-
Homo sapiens fragments of aggrecan
-
?

Synonyms

Synonyms Comment Organism
ADAMTS4
-
Homo sapiens
aggrecanase-1
-
Homo sapiens