Inhibitors | Comment | Organism | Structure |
---|---|---|---|
TIMP-2 | - |
Homo sapiens |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.4 | - |
peptide A13R | pH 7.5, 37°C | Homo sapiens | |
0.4 | - |
peptide A13P | pH 7.5, 37°C | Homo sapiens | |
0.6 | - |
peptide B74P | pH 7.5, 37°C | Homo sapiens | |
0.8 | - |
peptide B74R | pH 7.5, 37°C | Homo sapiens | |
1.3 | - |
peptide A13 | pH 7.5, 37°C | Homo sapiens | |
2.2 | - |
peptide A34 | pH 7.5, 37°C | Homo sapiens | |
2.2 | - |
peptide B74 | pH 7.5, 37°C | Homo sapiens | |
2.4 | - |
peptide B37 | pH 7.5, 37°C | Homo sapiens | |
3.2 | - |
peptide A21A | pH 7.5, 37°C | Homo sapiens | |
3.6 | - |
peptide A3 | pH 7.5, 37°C | Homo sapiens | |
4.4 | - |
peptide C9 | pH 7.5, 37°C | Homo sapiens | |
4.5 | - |
peptide B49 | pH 7.5, 37°C | Homo sapiens | |
6.4 | - |
peptide C9R | pH 7.5, 37°C | Homo sapiens | |
7.7 | - |
peptide A21 | pH 7.5, 37°C | Homo sapiens |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
additional information | Homo sapiens | important role in tumor angiogenesis | ? | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
human | - |
Purification (Comment) | Organism |
---|---|
catalytic domain | Homo sapiens |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
ephB1 + H2O | - |
Homo sapiens | ? | - |
? | |
additional information | important role in tumor angiogenesis | Homo sapiens | ? | - |
? | |
peptide A13 + H2O | - |
Homo sapiens | ? | - |
? | |
peptide A13P + H2O | - |
Homo sapiens | ? | - |
? | |
peptide A13R + H2O | - |
Homo sapiens | ? | - |
? | |
peptide A21 + H2O | - |
Homo sapiens | ? | - |
? | |
peptide A21A + H2O | - |
Homo sapiens | ? | - |
? | |
peptide A3 + H2O | - |
Homo sapiens | ? | - |
? | |
peptide A34 + H2O | - |
Homo sapiens | ? | - |
? | |
peptide B37 + H2O | - |
Homo sapiens | ? | - |
? | |
peptide B49 + H2O | - |
Homo sapiens | ? | - |
? | |
peptide B74 + H2O | - |
Homo sapiens | ? | - |
? | |
peptide B74P + H2O | - |
Homo sapiens | ? | - |
? | |
peptide B74R + H2O | - |
Homo sapiens | ? | - |
? | |
peptide C9 + H2O | - |
Homo sapiens | ? | - |
? | |
peptide C9R + H2O | - |
Homo sapiens | ? | - |
? |
Synonyms | Comment | Organism |
---|---|---|
gelatinase A | - |
Homo sapiens |
matrix metalloproteinase-2 | - |
Homo sapiens |
MMP-2 | - |
Homo sapiens |
Turnover Number Minimum [1/s] | Turnover Number Maximum [1/s] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
2 | 8 | peptide A13R | pH7.5, 37°C | Homo sapiens | |
61 | - |
peptide B74R | pH7.5, 37°C | Homo sapiens | |
105 | - |
peptide A13 | pH7.5, 37°C | Homo sapiens | |
124 | - |
peptide A21 | pH7.5, 37°C | Homo sapiens | |
202 | - |
peptide A34 | pH7.5, 37°C | Homo sapiens | |
204 | - |
peptide A13P | pH7.5, 37°C | Homo sapiens | |
264 | - |
peptide B74P | pH7.5, 37°C | Homo sapiens | |
353 | - |
peptide B37 | pH7.5, 37°C | Homo sapiens | |
400 | - |
peptide A3 | pH7.5, 37°C | Homo sapiens | |
510 | - |
peptide B49 | pH7.5, 37°C | Homo sapiens | |
601 | - |
peptide A21A | pH7.5, 37°C | Homo sapiens | |
622 | - |
peptide B74 | pH7.5, 37°C | Homo sapiens | |
740 | - |
peptide C9 | pH7.5, 37°C | Homo sapiens |