Inhibitors | Comment | Organism | Structure |
---|---|---|---|
Cbz-Leu-DL-Abu-CONH-(CH2)3-(4-methylpiperazin-1-yl) | - |
Sus scrofa | |
Cbz-Leu-DL-Abu-CONH-(CH2)3-2-methoxyadenin-9-yl | - |
Sus scrofa | |
Cbz-Leu-DL-Abu-CONH-(CH2)3-adenin-9-yl | - |
Sus scrofa | |
Cbz-Leu-DL-Abu-CONH-(CH2)3-cytosin-3-yl | - |
Sus scrofa | |
Cbz-Leu-DL-Abu-CONH-(CH2)3-morpholine | - |
Sus scrofa | |
CBZ-Leu-DL-Phe-CONH-(CH2)2-N-(CH3)2 | - |
Sus scrofa | |
CBZ-Leu-DL-Phe-CONH-(CH2)3-(4-methylpiperazin-1-yl) | - |
Sus scrofa | |
CBZ-Leu-DL-Phe-CONH-(CH2)3-2-methoxyadenin-9-yl | - |
Sus scrofa | |
CBZ-Leu-DL-Phe-CONH-(CH2)3-adenin-9-yl | best inhibitor | Sus scrofa | |
CBZ-Leu-DL-Phe-CONH-(CH2)3-cytosin-3-yl | - |
Sus scrofa | |
CBZ-Leu-DL-Phe-CONH-(CH2)3-N-(CH3)2 | - |
Sus scrofa |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Sus scrofa | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
kidney | - |
Sus scrofa | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
succinyl-Leu-Tyr-7-amido-4-methylcoumarin + H2O | - |
Sus scrofa | succinyl-Leu-Tyr + 7-amino-4-methylcoumarin | - |
? |
Synonyms | Comment | Organism |
---|---|---|
Cal II | - |
Sus scrofa |
calpain II | - |
Sus scrofa |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.000041 | - |
Cbz-Leu-DL-Abu-CONH-(CH2)3-morpholine | in 50 mM Tris-HCl, 50 mM NaCl, 1 mM EDTA, 1 mM EGTA, 0.1% CHAPS, pH 7.5, 10 mM dithiothreitol, 5 mM CaCl2, and less than 5% (v/v) DMSO, temperature not specified in the publication | Sus scrofa | |
0.000068 | - |
CBZ-Leu-DL-Phe-CONH-(CH2)3-adenin-9-yl | in 50 mM Tris-HCl, 50 mM NaCl, 1 mM EDTA, 1 mM EGTA, 0.1% CHAPS, pH 7.5, 10 mM dithiothreitol, 5 mM CaCl2, and less than 5% (v/v) DMSO, temperature not specified in the publication | Sus scrofa | |
0.00007 | - |
Cbz-Leu-DL-Abu-CONH-(CH2)3-adenin-9-yl | in 50 mM Tris-HCl, 50 mM NaCl, 1 mM EDTA, 1 mM EGTA, 0.1% CHAPS, pH 7.5, 10 mM dithiothreitol, 5 mM CaCl2, and less than 5% (v/v) DMSO, temperature not specified in the publication | Sus scrofa | |
0.000077 | - |
Cbz-Leu-DL-Abu-CONH-(CH2)3-2-methoxyadenin-9-yl | in 50 mM Tris-HCl, 50 mM NaCl, 1 mM EDTA, 1 mM EGTA, 0.1% CHAPS, pH 7.5, 10 mM dithiothreitol, 5 mM CaCl2, and less than 5% (v/v) DMSO, temperature not specified in the publication | Sus scrofa | |
0.000209 | - |
CBZ-Leu-DL-Phe-CONH-(CH2)3-2-methoxyadenin-9-yl | in 50 mM Tris-HCl, 50 mM NaCl, 1 mM EDTA, 1 mM EGTA, 0.1% CHAPS, pH 7.5, 10 mM dithiothreitol, 5 mM CaCl2, and less than 5% (v/v) DMSO, temperature not specified in the publication | Sus scrofa | |
0.000286 | - |
Cbz-Leu-DL-Abu-CONH-(CH2)3-(4-methylpiperazin-1-yl) | in 50 mM Tris-HCl, 50 mM NaCl, 1 mM EDTA, 1 mM EGTA, 0.1% CHAPS, pH 7.5, 10 mM dithiothreitol, 5 mM CaCl2, and less than 5% (v/v) DMSO, temperature not specified in the publication | Sus scrofa | |
0.000438 | - |
CBZ-Leu-DL-Phe-CONH-(CH2)3-cytosin-3-yl | in 50 mM Tris-HCl, 50 mM NaCl, 1 mM EDTA, 1 mM EGTA, 0.1% CHAPS, pH 7.5, 10 mM dithiothreitol, 5 mM CaCl2, and less than 5% (v/v) DMSO, temperature not specified in the publication | Sus scrofa | |
0.000844 | - |
CBZ-Leu-DL-Phe-CONH-(CH2)3-N-(CH3)2 | in 50 mM Tris-HCl, 50 mM NaCl, 1 mM EDTA, 1 mM EGTA, 0.1% CHAPS, pH 7.5, 10 mM dithiothreitol, 5 mM CaCl2, and less than 5% (v/v) DMSO, temperature not specified in the publication | Sus scrofa | |
0.00114 | - |
Cbz-Leu-DL-Abu-CONH-(CH2)3-cytosin-3-yl | in 50 mM Tris-HCl, 50 mM NaCl, 1 mM EDTA, 1 mM EGTA, 0.1% CHAPS, pH 7.5, 10 mM dithiothreitol, 5 mM CaCl2, and less than 5% (v/v) DMSO, temperature not specified in the publication | Sus scrofa | |
0.00352 | - |
CBZ-Leu-DL-Phe-CONH-(CH2)2-N-(CH3)2 | in 50 mM Tris-HCl, 50 mM NaCl, 1 mM EDTA, 1 mM EGTA, 0.1% CHAPS, pH 7.5, 10 mM dithiothreitol, 5 mM CaCl2, and less than 5% (v/v) DMSO, temperature not specified in the publication | Sus scrofa | |
0.00636 | - |
CBZ-Leu-DL-Phe-CONH-(CH2)3-(4-methylpiperazin-1-yl) | in 50 mM Tris-HCl, 50 mM NaCl, 1 mM EDTA, 1 mM EGTA, 0.1% CHAPS, pH 7.5, 10 mM dithiothreitol, 5 mM CaCl2, and less than 5% (v/v) DMSO, temperature not specified in the publication | Sus scrofa |