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Literature summary for 3.4.22.16 extracted from

  • Brguljan, P.M.; Turk, V.; Nina, C.; Brzin, J.; Krizaj, I.; Popovic, T.
    Human brain cathepsin H as a neuropeptide and bradykinin metabolizing enzyme (2003), Peptides, 24, 1977-1984.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
cystatin C, full-length
-
Homo sapiens
cystatin C, truncated form deletion of 10 N-terminal amino acids Homo sapiens

Molecular Weight [Da]

Molecular Weight [Da] Molecular Weight Maximum [Da] Comment Organism
30000
-
x * 30000, SDS-PAGE Homo sapiens

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
brain
-
Homo sapiens
-

Specific Activity [micromol/min/mg]

Specific Activity Minimum [µmol/min/mg] Specific Activity Maximum [µmol/min/mg] Comment Organism
2
-
-
Homo sapiens

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
alpha-neoendorphin + H2O preferentially aminopeptidase activity, endoeptidase activity after prolonged incubation Homo sapiens ?
-
?
bradykinin + H2O no aminopeptidase activity, endopeptidase activity after prolonged incubation Homo sapiens ?
-
?
demorphin + H2O no aminopeptidase activity, endopeptidase activity after prolonged incubation Homo sapiens ?
-
?
dynorphin(1-13) + H2O preferentially aminopeptidase activity, endoeptidase activity after prolonged incubation Homo sapiens ?
-
?
dynorphin(1-6) + H2O preferentially aminopeptidase activity, endoeptidase activity after prolonged incubation Homo sapiens ?
-
?
Leu-enkephalin + H2O preferentially aminopeptidase activity, endoeptidase activity after prolonged incubation Homo sapiens ?
-
?
Lys-bradykinin + H2O preferentially aminopeptidase activity, endoeptidase activity after prolonged incubation Homo sapiens ?
-
?
neurotensin + H2O no aminopeptidase activity, endopeptidase activity after prolonged incubation Homo sapiens ?
-
?

Subunits

Subunits Comment Organism
? x * 30000, SDS-PAGE Homo sapiens

Ki Value [mM]

Ki Value [mM] Ki Value maximum [mM] Inhibitor Comment Organism Structure
0.000000071
-
cystatin C, full-length 25°C, pH 7.0 Homo sapiens
0.00000032
-
cystatin C, truncated form 25°C, pH 7.0 Homo sapiens

pI Value

Organism Comment pI Value Maximum pI Value
Homo sapiens and minor band at 6.1, isoelectric focusing 6.8 6.3