Cloned (Comment) | Organism |
---|---|
expressed in insect cell/baculovirus expression system | Homo sapiens |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
8,8'-paepalantine dimer | potent competitive inhibitor | Homo sapiens | |
paepalantine | - |
Homo sapiens | |
vioxanthin | potent competitive inhibitor | Homo sapiens |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.004 | - |
Abz-KLRSSKQ-EDDnp | pH and temperature not specified in the publication | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
Abz-KLRSSKQ-EDDnp + H2O | - |
Homo sapiens | ? | - |
? | |
additional information | no activity with Abz-KLYSSKQ-EDDnp | Homo sapiens | ? | - |
? |
Synonyms | Comment | Organism |
---|---|---|
kallikrein 5 | - |
Homo sapiens |
KLK5 | - |
Homo sapiens |
Turnover Number Minimum [1/s] | Turnover Number Maximum [1/s] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
8.5 | - |
Abz-KLRSSKQ-EDDnp | pH and temperature not specified in the publication | Homo sapiens |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.0229 | - |
vioxanthin | pH and temperature not specified in the publication | Homo sapiens | |
0.0244 | - |
8,8'-paepalantine dimer | pH and temperature not specified in the publication | Homo sapiens | |
0.0475 | - |
paepalantine | pH and temperature not specified in the publication | Homo sapiens |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.0537 | - |
pH and temperature not specified in the publication | Homo sapiens | vioxanthin | |
0.0729 | - |
pH and temperature not specified in the publication | Homo sapiens | 8,8'-paepalantine dimer | |
0.3674 | - |
pH and temperature not specified in the publication | Homo sapiens | paepalantine |
kcat/KM Value [1/mMs-1] | kcat/KM Value Maximum [1/mMs-1] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
2125 | - |
Abz-KLRSSKQ-EDDnp | pH and temperature not specified in the publication | Homo sapiens |