Application | Comment | Organism |
---|---|---|
medicine | involved in host cell invasion, important target for drug design | Escherichia coli |
Cloned (Comment) | Organism |
---|---|
overexpressed in Escherichia coli JM83 | Escherichia coli |
Protein Variants | Comment | Organism |
---|---|---|
Y452F | site-specific mutagenesis | Escherichia coli |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
acetyl-Thr-Arg-Arg | - |
Escherichia coli | |
benzamidine | - |
Escherichia coli |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.0048 | - |
2-aminobenzoyl-Thr-Arg-Arg Phe(NO2)-Ser-Leu-NH2 | pH 8.0, 25°C, 3 mM | Escherichia coli | |
0.014 | - |
2-aminobenzoyl-Thr-Arg-Arg Phe(NO2)-Ser-Leu-NH2 | pH 8.0, 15°C, 1 M | Escherichia coli | |
0.024 | - |
2-aminobenzoyl-Thr-Arg-Arg Phe(NO2)-Ser-Leu-NH2 | pH 8.0, 25°C | Escherichia coli | |
0.0298 | - |
2-aminobenzoyl-Thr-Arg Cit-Phe(NO2)-Ser-Leu-NH2 | pH 8.0, 25°C | Escherichia coli | |
0.0379 | - |
2-aminobenzoyl-Thr-Arg-Arg Phe(NO2)-Ser-Leu-NH2 | pH 8.0, 35°C | Escherichia coli | |
0.08 | - |
2-aminobenzoyl-Thr-Cit-Arg Phe(NO2)-Ser-Leu-NH2 | pH 8.0, 25°C, 1 M | Escherichia coli | |
0.083 | - |
2-aminobenzoyl-Thr-Arg-Arg Phe(NO2)-Ser-Leu-NH2 | pH 8.0, 25°C | Escherichia coli |
Metals/Ions | Comment | Organism | Structure |
---|---|---|---|
Ca2+ | activation at 5-10 mM CaCl2 | Escherichia coli |
Molecular Weight [Da] | Molecular Weight Maximum [Da] | Comment | Organism |
---|---|---|---|
81860 | - |
amino acid sequence | Escherichia coli |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
additional information | Escherichia coli | involved in host cell invasion | ? | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Escherichia coli | - |
- |
- |
Purification (Comment) | Organism |
---|---|
- |
Escherichia coli |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
2-aminobenzoyl-Thr-Arg Cit-Phe(NO2)-Ser-Leu-NH2 + H2O | - |
Escherichia coli | ? | - |
? | |
2-aminobenzoyl-Thr-Arg-Arg Phe(NO2)-Ser-Leu-NH2 + H2O | - |
Escherichia coli | ? | - |
? | |
2-aminobenzoyl-Thr-Cit-Arg Phe(NO2)-Ser-Leu-NH2 + H2O | - |
Escherichia coli | ? | - |
? | |
2-aminobenzoyl-Thr-Cit-Cit-Phe(NO2)-Ser-Leu-NH2 + H2O | - |
Escherichia coli | ? | - |
? | |
benzoyl-Arg-Et + H2O | - |
Escherichia coli | ? | - |
? | |
benzoyl-Arg-NH2 + H2O | - |
Escherichia coli | ? | - |
? | |
benzoyl-citrulline-Et + H2O | - |
Escherichia coli | ? | - |
? | |
benzyloxycarbonyl-Arg-Arg-7-(4-methylcoumaryl)amide + H2O | - |
Escherichia coli | ? | - |
? | |
additional information | specific for substrates with a pair of basic residues at positions P1 and P2 | Escherichia coli | ? | - |
? | |
additional information | involved in host cell invasion | Escherichia coli | ? | - |
? | |
Nalpha-benzoyl-L-Arg 2-naphthylamide + H2O | - |
Escherichia coli | Nalpha-benzoyl-L-Arg + 2-naphthylamine | - |
? |
Temperature Optimum [°C] | Temperature Optimum Maximum [°C] | Comment | Organism |
---|---|---|---|
25 | - |
the abnormally low temperature optimum may be caused by the disruption of the hydrogen bond formed between the enzyme and the NH group of the scissile peptide bond | Escherichia coli |
Turnover Number Minimum [1/s] | Turnover Number Maximum [1/s] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
294 | - |
2-aminobenzoyl-Thr-Arg Cit-Phe(NO2)-Ser-Leu-NH2 | pH 8.0, 25°C | Escherichia coli | |
516 | - |
2-aminobenzoyl-Thr-Arg-Arg Phe(NO2)-Ser-Leu-NH2 | pH 8.0, 15°C, 1 M | Escherichia coli | |
1218 | - |
2-aminobenzoyl-Thr-Cit-Arg Phe(NO2)-Ser-Leu-NH2 | pH 8.0, 25°C | Escherichia coli | |
1220 | - |
2-aminobenzoyl-Thr-Cit-Arg Phe(NO2)-Ser-Leu-NH2 | pH 8.0, 25°C | Escherichia coli | |
1260 | - |
2-aminobenzoyl-Thr-Arg-Arg Phe(NO2)-Ser-Leu-NH2 | pH 8.0, 25°C, 3 mM | Escherichia coli | |
1390 | - |
2-aminobenzoyl-Thr-Arg-Arg Phe(NO2)-Ser-Leu-NH2 | pH 8.0, 25°C | Escherichia coli | |
1392 | - |
2-aminobenzoyl-Thr-Arg-Arg Phe(NO2)-Ser-Leu-NH2 | pH 8.0, 25°C | Escherichia coli | |
1416 | - |
2-aminobenzoyl-Thr-Arg-Arg Phe(NO2)-Ser-Leu-NH2 | pH 8.0, 35°C | Escherichia coli | |
1420 | - |
2-aminobenzoyl-Thr-Arg-Arg Phe(NO2)-Ser-Leu-NH2 | pH 8.0, 35°C | Escherichia coli |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
8 | - |
- |
Escherichia coli |
pH Minimum | pH Maximum | Comment | Organism |
---|---|---|---|
6.5 | 9.5 | - |
Escherichia coli |