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Literature summary for 3.4.21.75 extracted from

  • Liu, Z.X.; Fei, H.; Chi, C.W.
    Two engineered eglin c mutants potently and selectively inhibiting kexin or furin (2004), FEBS Lett., 556, 116-120.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
eglin c Arg replaced with Asp at P3
-
Saccharomyces cerevisiae
eglin c mutant D42R
-
Saccharomyces cerevisiae
eglin c mutant L45R
-
Saccharomyces cerevisiae
eglin variant M1 RVTR
-
Saccharomyces cerevisiae
eglin variant M2 RVKR
-
Saccharomyces cerevisiae
eglin variant M3 RVTRDERY
-
Saccharomyces cerevisiae
eglin variant M4 RVTRDRRY
-
Saccharomyces cerevisiae
eglin variant M5 RVTRDLDY
-
Saccharomyces cerevisiae
eglin variant M6 RVTRDLRR
-
Saccharomyces cerevisiae
eglin variant M7 RVTRDLRE
-
Saccharomyces cerevisiae
eglin variant M8 RVTRDARY
-
Saccharomyces cerevisiae

Localization

Localization Comment Organism GeneOntology No. Textmining
Golgi apparatus trans Golgi network Saccharomyces cerevisiae 5794
-

Organism

Organism UniProt Comment Textmining
Saccharomyces cerevisiae
-
yeast
-

Ki Value [mM]

Ki Value [mM] Ki Value maximum [mM] Inhibitor Comment Organism Structure
0.0000016
-
eglin variant M2 RVKR pH 7.5, 37°C Saccharomyces cerevisiae
0.0000078
-
eglin variant M5 RVTRDLDY pH 7.5, 37°C Saccharomyces cerevisiae
0.0000078
-
eglin c mutant Arg replaced with Asp at P3 pH 7.5, 37°C Saccharomyces cerevisiae
0.00002
-
eglin variant M8 RVTRDARY pH 7.5, 37°C Saccharomyces cerevisiae
0.000023
-
eglin c mutant L45R pH 7.5, 37°C Saccharomyces cerevisiae
0.000023
-
eglin c mutant D42R pH 7.5, 37°C Saccharomyces cerevisiae
0.000023
-
eglin variant M1 RVTR pH 7.5, 37°C Saccharomyces cerevisiae
0.000039
-
eglin variant M7 RVTRDLRE pH 7.5, 37°C Saccharomyces cerevisiae
0.000047
-
eglin variant M6 RVTRDLRR pH 7.5, 37°C Saccharomyces cerevisiae
0.0003
-
eglin variant M4 RVTRDRRY pH 7.5, 37°C Saccharomyces cerevisiae
0.00092
-
eglin variant M3 RVTRDERY pH 7.5, 37°C Saccharomyces cerevisiae