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Literature summary for 3.4.21.73 extracted from

  • Bergstrom, R.C.; Coombs, G.S.; Ye, S.; Madison, E.L.; Goldsmith, E.J.; Corey, D.R.
    Binding of nonphysiological protein and peptide substrates to proteases: differences between urokinase-type plasminogen activator and trypsin and contributions to the evolution of regulated proteolysis (2003), Biochemistry, 42, 5395-5402.
    View publication on PubMed

Protein Variants

Protein Variants Comment Organism
S195A/C122S/N145D inactive variant Homo sapiens

KM Value [mM]

KM Value [mM] KM Value Maximum [mM] Substrate Comment Organism Structure
0.014
-
PFGRSA pH 7.5, 37°C, protein substrate Homo sapiens
0.03
-
HYGRSA pH 7.5, 37°C, protein substrate Homo sapiens
0.052
-
GSGRSA pH 7.5, 37°C, protein substrate Homo sapiens
0.13
-
QRGRSA pH 7.5, 37°C, protein substrate Homo sapiens
0.13
-
YGAKAY pH 7.5, 37°C, protein substrate Homo sapiens
0.6
-
GSGRSA pH 7.5, 37°C, peptide substrate Homo sapiens
2.18
-
QRGRSA pH 7.5, 37°C, peptide substrate Homo sapiens
2.2
-
PFGRSA pH 7.5, 37°C, peptide substrate Homo sapiens
2.3
-
YGAKAY pH 7.5, 37°C, peptide substrate Homo sapiens
3.8
-
HYGRSA pH 7.5, 37°C, peptide substrate Homo sapiens

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
human
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
GSGRSA + H2O
-
Homo sapiens GSGR + Ser-Ala
-
?
HYGRSA + H2O
-
Homo sapiens HYGR + Ser-Ala
-
?
PFGRSA + H2O
-
Homo sapiens PFGR + Ser-Ala
-
?
QRGRSA + H2O
-
Homo sapiens QRGR + Ser-Ala
-
?
YGAKAY + H2O
-
Homo sapiens YGAK + Ala-Tyr
-
?

Synonyms

Synonyms Comment Organism
Urokinase-type plasminogen activator
-
Homo sapiens