Inhibitors | Comment | Organism | Structure |
---|---|---|---|
2,2,4,7-tetramethyl-6-[2-(4-methylphenyl)[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]-1,2,3,4-tetrahydroquinoline | 89% activity at 0.03 mM | Homo sapiens | |
6-[2-(4-chlorophenyl)[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]-2,2,4,7-tetramethyl-1,2,3,4-tetrahydroquinoline | 16% activity at 0.005 mM; 35% activity at 0.03 mM; 63% activity at 0.001 mM; 67% activity at 0.03 mM; 76% activity at 0.005 mM; 82% activity at 0.03 mM; 85% activity at 0.005 mM; 87% activity at 0.03 mM; 8% activity at 0.005 mM; 94% activity at 0.03 mM | Homo sapiens | |
additional information | not inhibited by VGY-000058 | Homo sapiens | |
N-(2,4-dichlorophenyl)-4-(2,2,4,7-tetramethyl-1,2,3,4-tetrahydroquinolin-6-yl)pyrimidin-2-amine | 1% activity at 0.03 mM | Homo sapiens | |
rivaroxaban | - |
Homo sapiens | |
VGY-000010 | - |
Homo sapiens | |
VGY-000014 | - |
Homo sapiens | |
VGY-000046 | - |
Homo sapiens | |
VGY-000049 | - |
Homo sapiens | |
VGY-000060 | - |
Homo sapiens | |
VGY-000063 | - |
Homo sapiens | |
VGY-000073 | - |
Homo sapiens | |
VGY-0006201 | - |
Homo sapiens | |
VGY-0006208 | - |
Homo sapiens | |
VGY-0006212 | - |
Homo sapiens | |
VGY-0224586 | - |
Homo sapiens | |
VGY-0224865 | - |
Homo sapiens | |
VGY-0224867 | - |
Homo sapiens | |
VGY-0224887 | - |
Homo sapiens | |
VGY-0224908 | - |
Homo sapiens | |
VGY-0224909 | - |
Homo sapiens | |
VGY-0224918 | - |
Homo sapiens | |
VGY-0224933 | - |
Homo sapiens | |
VGY-0224945 | - |
Homo sapiens | |
VGY-0224950 | - |
Homo sapiens | |
VGY-0224963 | - |
Homo sapiens | |
VGY-0224989 | - |
Homo sapiens | |
VGY-0225108 | - |
Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | P00742 | - |
- |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
Z-D-Arg-Gly-Arg-4-nitroanilide + H2O | i.e S2765 | Homo sapiens | Z-D-Arg-Gly-Arg + 4-nitroaniline | - |
? |
Synonyms | Comment | Organism |
---|---|---|
FXa | - |
Homo sapiens |