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Literature summary for 3.4.21.59 extracted from

  • Jiang, Q.Q.; Bartsch, L.; Sicking, W.; Wich, P.R.; Heider, D.; Hoffmann, D.; Schmuck, C.
    A new approach to inhibit human beta-tryptase by protein surface binding of four-armed peptide ligands with two different sets of arms (2013), Org. Biomol. Chem., 11, 1631-1639.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
leech-derived tryptase inhibitor nanomolar inhibitor Homo sapiens
MCoTI-II derived miniprotein nanomolar inhibitor Homo sapiens

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
tosyl-Gly-L-Pro-L-Arg-7-amido-4-methylcoumarin + H2O
-
Homo sapiens tosyl-Gly-L-Pro-L-Arg + 7-amino-4-methylcoumarin
-
?

Synonyms

Synonyms Comment Organism
beta-tryptase
-
Homo sapiens