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Literature summary for 3.4.21.22 extracted from

  • Sullenger, B.; Woodruff, R.; Monroe, D.M.
    Potent anticoagulant aptamer directed against factor IXa blocks macromolecular substrate interaction (2012), J. Biol. Chem., 287, 12779-12786.
    View publication on PubMedView publication on EuropePMC

Activating Compound

Activating Compound Comment Organism Structure
Factor VIIIa
-
Homo sapiens
tissue factor
-
Homo sapiens

Inhibitors

Inhibitors Comment Organism Structure
additional information aptamer 9.3t blocks the activity of factor IXa-factor VIIIa complex Homo sapiens

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
Factor X + H2O Homo sapiens
-
Factor Xa + ?
-
?

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-

Purification (Commentary)

Purification (Comment) Organism
DEAE-Sepharose column chromatography and HiTrap Q column chromatography Homo sapiens

Source Tissue

Source Tissue Comment Organism Textmining
blood plasma
-
Homo sapiens
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
D-Leu-Phe-Gly-Arg-4-nitroanilide + H2O
-
Homo sapiens D-Leu-Phe-Gly-Arg + 4-nitroaniline
-
?
Factor X + H2O
-
Homo sapiens Factor Xa + ?
-
?

Synonyms

Synonyms Comment Organism
factor IXa
-
Homo sapiens
FIXa
-
Homo sapiens