Activating Compound | Comment | Organism | Structure |
---|---|---|---|
dithiothreitol | absolute requirement for maintenance of activity | Homo sapiens |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
amastatin | - |
Homo sapiens | |
Arphamenine B | - |
Homo sapiens | |
chymostatin | - |
Homo sapiens | |
Elastinal | - |
Homo sapiens | |
leupeptin | - |
Homo sapiens | |
NEM | - |
Homo sapiens |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.08 | - |
pyroglutamate-4-methylcoumarin 7-amide | - |
Homo sapiens |
Metals/Ions | Comment | Organism | Structure |
---|---|---|---|
additional information | maximal activity in absence of divalent cations | Homo sapiens |
Molecular Weight [Da] | Molecular Weight Maximum [Da] | Comment | Organism |
---|---|---|---|
22000 | - |
gel filtration | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Purification (Comment) | Organism |
---|---|
- |
Homo sapiens |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
skeletal muscle | quadriceps muscle | Homo sapiens | - |
Specific Activity Minimum [µmol/min/mg] | Specific Activity Maximum [µmol/min/mg] | Comment | Organism |
---|---|---|---|
1.093 | - |
- |
Homo sapiens |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
luliberin + H2O | - |
Homo sapiens | pyroglutamate + His-Trp-Ser-Tyr-Gly-Leu-Arg-Pro-Gly-NH2 | - |
? | |
neurotensin + H2O | - |
Homo sapiens | pyroglutamate + Leu-Tyr-Glu-Asn-Lys-Pro-Ag-Arg-Pro-Tyr-Ile-Leu | - |
? | |
pyroglutamyl-4-methylcoumarin 7-amide + H2O | - |
Homo sapiens | pyroglutamate + 7-amino-4-methylcoumarin | - |
? | |
thyroliberin + H2O | - |
Homo sapiens | pyroglutamate + His-Pro-NH2 | - |
? |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
8.5 | - |
- |
Homo sapiens |
pH Minimum | pH Maximum | Comment | Organism |
---|---|---|---|
7 | 9.5 | 50% of maximal activity at pH 7 and at pH 9.5 | Homo sapiens |