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Literature summary for 3.4.15.1 extracted from

  • Ceconi, C.; Francolini, G.; Olivares, A.; Comini, L.; Bachetti, T.; Ferrari, R.
    Angiotensin-converting enzyme (ACE) inhibitors have different selectivity for bradykinin binding sites of human somatic ACE (2007), Eur. J. Pharmacol., 577, 1-6.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
angiotensin I
-
Homo sapiens
bradykinin
-
Homo sapiens
enalaprilat
-
Homo sapiens
perindoprilat
-
Homo sapiens
quinaprilat
-
Homo sapiens
ramiprilat
-
Homo sapiens
trandolaprilat
-
Homo sapiens

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
HUVEC cell
-
Homo sapiens
-

Ki Value [mM]

Ki Value [mM] Ki Value maximum [mM] Inhibitor Comment Organism Structure
0.00000035
-
quinaprilat
-
Homo sapiens
0.00000057
-
trandolaprilat
-
Homo sapiens
0.00000076
-
ramiprilat
-
Homo sapiens
0.00000105
-
perindoprilat
-
Homo sapiens
0.000001278
-
bradykinin
-
Homo sapiens
0.00000194
-
enalaprilat
-
Homo sapiens
0.000002747
-
angiotensin I
-
Homo sapiens