Inhibitors | Comment | Organism | Structure |
---|---|---|---|
PF-00734200 | potent, competitive DPP-IV inhibitor, complete inhibition of DPP-IV for over 24 h after treatment with one single dose of 300 mg PF-00734200 | Homo sapiens |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
glucagon-like peptide 1 + H2O | Homo sapiens | - |
? | - |
? | |
glucose-dependent insulinotropic peptide + H2O | Homo sapiens | - |
? | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
blood plasma | - |
Homo sapiens | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
glucagon-like peptide 1 + H2O | - |
Homo sapiens | ? | - |
? | |
glucose-dependent insulinotropic peptide + H2O | - |
Homo sapiens | ? | - |
? | |
Gly-L-Pro-7-amido-4-methylcoumarin + H2O | - |
Homo sapiens | Gly-L-Pro + 7-amino-4-methylcoumarin | - |
? |
Synonyms | Comment | Organism |
---|---|---|
dipeptidyl peptidase-IV | - |
Homo sapiens |
DPP-IV | - |
Homo sapiens |