Activating Compound | Comment | Organism | Structure |
---|---|---|---|
TGF-beta1 | activates aminopeptidase activity | Rattus norvegicus |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
actinonin | 40% inhibition at 0.0003 mM, independent on TGF-beta1 activation | Rattus norvegicus | |
amastatin | 50-70% inhibition at 0.0003 mM, dependent on TGF-beta1 activation | Rattus norvegicus | |
arphamenine A | aminopeptidase B-specific inhibitor | Rattus norvegicus | |
bestatin | strong inhibition | Rattus norvegicus | |
L-Arg-2-naphthylamide | competitive inhibition of hydrolysis of L-Ala-2-naphthylamide, no inhibition vice versa | Rattus norvegicus | |
leuhistin | 40% inhibition at 0.0003 mM, independent on TGF-beta1 activation | Rattus norvegicus | |
additional information | no or poor inhibition of L-Arg-2-naphthylamide hydrolysis by puromycin at 1 mM, aprotinin, pepstatin A, E64, chymostatin, imipramine, phosphoramidon, lisinopril, and apstatin | Rattus norvegicus |
Localization | Comment | Organism | GeneOntology No. | Textmining |
---|---|---|---|---|
cytosol | - |
Rattus norvegicus | 5829 | - |
extracellular | - |
Rattus norvegicus | - |
- |
membrane | - |
Rattus norvegicus | 16020 | - |
additional information | subcellular localization, overview | Rattus norvegicus | - |
- |
Metals/Ions | Comment | Organism | Structure |
---|---|---|---|
Cl- | activates | Rattus norvegicus |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Rattus norvegicus | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
fibroblast | cardiac, ventricular | Rattus norvegicus | - |
heart | cardiac ventricular fibroblastic cell | Rattus norvegicus | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
L-Ala-2-naphthylamide + H2O | - |
Rattus norvegicus | L-Ala + 2-naphthylamine | - |
? | |
L-Ala-4-nitroanilide + H2O | - |
Rattus norvegicus | L-Ala + 4-nitroaniline | - |
? | |
L-Arg-2-naphthylamide + H2O | - |
Rattus norvegicus | L-Arg + 2-naphthylamine | - |
? | |
L-Arg-4-nitroanilide + H2O | - |
Rattus norvegicus | L-Arg + 4-nitroaniline | - |
? | |
L-Lys-2-naphthylamide + H2O | - |
Rattus norvegicus | L-Lys + 2-naphthylamine | - |
? | |
L-Lys-4-nitroanilide + H2O | - |
Rattus norvegicus | L-Lys + 4-nitroaniline | - |
? |
Synonyms | Comment | Organism |
---|---|---|
Ap-B | - |
Rattus norvegicus |
Arg-AP | - |
Rattus norvegicus |
arginine-aminopeptidase | - |
Rattus norvegicus |
Temperature Optimum [°C] | Temperature Optimum Maximum [°C] | Comment | Organism |
---|---|---|---|
37 | - |
assay at | Rattus norvegicus |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
7.2 | - |
assay at | Rattus norvegicus |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
additional information | - |
additional information | - |
Rattus norvegicus |