Inhibitors | Comment | Organism | Structure |
---|---|---|---|
1-methyl-N-[3-(1H-tetrazol-5-yl)phenyl]-1H-indole-6-sulfonamide | - |
Cricetulus griseus | |
2,4,5-trichloro-N-[3-(1H-tetrazol-5-yl)phenyl]benzenesulfonamide | - |
Cricetulus griseus | |
3,4-dichloro-N-[3-(1H-tetrazol-5-yl)phenyl]benzenesulfonamide | - |
Cricetulus griseus | |
3,4-dimethyl-N-[3-(1H-tetrazol-5-yl)phenyl]benzenesulfonamide | - |
Cricetulus griseus | |
3-([(4-bromo-5-chlorothiophen-2-yl)sulfonyl]amino)-N-methylbenzamide | - |
Cricetulus griseus | |
4,5-dichloro-N-[3-(1H-tetrazol-5-yl)phenyl]thiophene-2-sulfonamide | - |
Cricetulus griseus | |
4-bromo-2,6-difluoro-N-[3-(1H-tetrazol-5-yl)phenyl]benzenesulfonamide | - |
Cricetulus griseus | |
4-bromo-2-fluoro-N-[3-(1H-tetrazol-5-yl)phenyl]benzenesulfonamide | - |
Cricetulus griseus | |
4-bromo-5-chloro-N-methyl-N-[3-(1H-tetrazol-5-yl)phenyl]thiophene-2-sulfonamide | - |
Cricetulus griseus | |
4-bromo-5-chloro-N-[3-(1-methyl-1H-tetrazol-5-yl)phenyl]thiophene-2-sulfonamide | - |
Cricetulus griseus | |
4-bromo-5-chloro-N-[3-(1H-tetrazol-5-yl)phenyl]thiophene-2-carboxamide | - |
Cricetulus griseus | |
4-bromo-5-chloro-N-[3-(1H-tetrazol-5-yl)phenyl]thiophene-2-sulfonamide | - |
Cricetulus griseus | |
7-chloro-N-[3-(1H-tetrazol-5-yl)phenyl]-1,3-dihydro-2,1,3-benzoxadiazole-4-sulfonamide | - |
Cricetulus griseus | |
N-[3-(1H-tetrazol-5-yl)phenyl]-1-benzothiophene-2-sulfonamide | - |
Cricetulus griseus | |
N-[3-(1H-tetrazol-5-yl)phenyl]-2-benzothiophene-4-sulfonamide | - |
Cricetulus griseus | |
N-[3-(1H-tetrazol-5-yl)phenyl]benzenesulfonamide | - |
Cricetulus griseus | |
N-[3-(1H-tetrazol-5-yl)phenyl]biphenyl-4-sulfonamide | - |
Cricetulus griseus | |
N-[3-(1H-tetrazol-5-yl)phenyl]pyridine-3-sulfonamide | - |
Cricetulus griseus | |
N-[3-(1H-tetrazol-5-yl)phenyl]thiophene-2-sulfonamide | - |
Cricetulus griseus |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Cricetulus griseus | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
CHO cell | - |
Cricetulus griseus | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
L-Leu-4-nitroanilide + H2O | - |
Cricetulus griseus | L-Leu + 4-nitroaniline | - |
? |
Synonyms | Comment | Organism |
---|---|---|
insulin-regulated aminopeptidase | - |
Cricetulus griseus |
IRAP | - |
Cricetulus griseus |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
7.4 | - |
assay at | Cricetulus griseus |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.0011 | - |
pH 7.4, temperature not specified in the publication | Cricetulus griseus | 3,4-dichloro-N-[3-(1H-tetrazol-5-yl)phenyl]benzenesulfonamide | |
0.0013 | - |
pH 7.4, temperature not specified in the publication | Cricetulus griseus | 7-chloro-N-[3-(1H-tetrazol-5-yl)phenyl]-1,3-dihydro-2,1,3-benzoxadiazole-4-sulfonamide | |
0.0016 | - |
pH 7.4, temperature not specified in the publication | Cricetulus griseus | 4-bromo-2-fluoro-N-[3-(1H-tetrazol-5-yl)phenyl]benzenesulfonamide | |
0.0018 | - |
pH 7.4, temperature not specified in the publication | Cricetulus griseus | 4,5-dichloro-N-[3-(1H-tetrazol-5-yl)phenyl]thiophene-2-sulfonamide | |
0.0021 | - |
pH 7.4, temperature not specified in the publication | Cricetulus griseus | 4-bromo-5-chloro-N-[3-(1H-tetrazol-5-yl)phenyl]thiophene-2-sulfonamide | |
0.0029 | - |
pH 7.4, temperature not specified in the publication | Cricetulus griseus | 2,4,5-trichloro-N-[3-(1H-tetrazol-5-yl)phenyl]benzenesulfonamide | |
0.0031 | - |
pH 7.4, temperature not specified in the publication | Cricetulus griseus | 3,4-dimethyl-N-[3-(1H-tetrazol-5-yl)phenyl]benzenesulfonamide | |
0.0079 | - |
pH 7.4, temperature not specified in the publication | Cricetulus griseus | 4-bromo-2,6-difluoro-N-[3-(1H-tetrazol-5-yl)phenyl]benzenesulfonamide | |
0.016 | - |
pH 7.4, temperature not specified in the publication | Cricetulus griseus | N-[3-(1H-tetrazol-5-yl)phenyl]-1-benzothiophene-2-sulfonamide | |
0.022 | - |
pH 7.4, temperature not specified in the publication | Cricetulus griseus | 1-methyl-N-[3-(1H-tetrazol-5-yl)phenyl]-1H-indole-6-sulfonamide | |
0.039 | - |
pH 7.4, temperature not specified in the publication | Cricetulus griseus | N-[3-(1H-tetrazol-5-yl)phenyl]-2-benzothiophene-4-sulfonamide | |
0.044 | - |
pH 7.4, temperature not specified in the publication | Cricetulus griseus | N-[3-(1H-tetrazol-5-yl)phenyl]biphenyl-4-sulfonamide | |
0.058 | - |
pH 7.4, temperature not specified in the publication | Cricetulus griseus | 4-bromo-5-chloro-N-methyl-N-[3-(1H-tetrazol-5-yl)phenyl]thiophene-2-sulfonamide | |
0.067 | - |
pH 7.4, temperature not specified in the publication | Cricetulus griseus | 4-bromo-5-chloro-N-[3-(1H-tetrazol-5-yl)phenyl]thiophene-2-carboxamide | |
0.125 | - |
pH 7.4, temperature not specified in the publication | Cricetulus griseus | 4-bromo-5-chloro-N-[3-(1-methyl-1H-tetrazol-5-yl)phenyl]thiophene-2-sulfonamide | |
0.125 | - |
pH 7.4, temperature not specified in the publication | Cricetulus griseus | 3-([(4-bromo-5-chlorothiophen-2-yl)sulfonyl]amino)-N-methylbenzamide | |
0.125 | - |
pH 7.4, temperature not specified in the publication | Cricetulus griseus | N-[3-(1H-tetrazol-5-yl)phenyl]thiophene-2-sulfonamide | |
0.125 | - |
pH 7.4, temperature not specified in the publication | Cricetulus griseus | N-[3-(1H-tetrazol-5-yl)phenyl]benzenesulfonamide | |
0.125 | - |
pH 7.4, temperature not specified in the publication | Cricetulus griseus | N-[3-(1H-tetrazol-5-yl)phenyl]pyridine-3-sulfonamide |