Inhibitors | Comment | Organism | Structure |
---|---|---|---|
amastatin | - |
Homo sapiens | |
amastatin | - |
Oryctolagus cuniculus | |
D-Arg-L-Lys-[Hyp3, CpG5, D-Tic7, CpG8]des-Arg9-bradykinin | competitive to L-Ala-4-nitroanilide, additionally inhibitory to kinin B1 receptor | Homo sapiens | |
D-Arg-L-Lys-[Hyp3, CpG5, D-Tic7, CpG8]des-Arg9-bradykinin | competitive to L-Ala-4-nitroanilide, additionally inhibitory to kinin B1 receptor | Oryctolagus cuniculus | |
L-Lys-L-Lys-[Hyp3, CpG5, D-Tic7, CpG8]des-Arg9-bradykinin | competitive to L-Ala-4-nitroanilide | Homo sapiens | |
L-Lys-L-Lys-[Hyp3, CpG5, D-Tic7, CpG8]des-Arg9-bradykinin | competitive to L-Ala-4-nitroanilide | Oryctolagus cuniculus |
Localization | Comment | Organism | GeneOntology No. | Textmining |
---|---|---|---|---|
membrane | - |
Homo sapiens | 16020 | - |
membrane | - |
Oryctolagus cuniculus | 16020 | - |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Oryctolagus cuniculus | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
artery | arterial smooth muscle | Homo sapiens | - |
artery | arterial smooth muscle | Oryctolagus cuniculus | - |
smooth muscle | arterial smooth muscle | Homo sapiens | - |
smooth muscle | arterial smooth muscle | Oryctolagus cuniculus | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
L-Ala-4-nitroanilide + H2O | - |
Homo sapiens | L-Ala + 4-nitroaniline | - |
? | |
L-Ala-4-nitroanilide + H2O | - |
Oryctolagus cuniculus | L-Ala + 4-nitroaniline | - |
? | |
L-Lys-L-Lys-[Hyp3, CpG5, D-Tic7, CpG8]des-Arg9-bradykinin + H2O | i.e.B-9958 | Homo sapiens | ? | - |
? | |
L-Lys-L-Lys-[Hyp3, CpG5, D-Tic7, CpG8]des-Arg9-bradykinin + H2O | i.e.B-9958 | Oryctolagus cuniculus | ? | - |
? |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.00086 | - |
D-Arg-L-Lys-[Hyp3, CpG5, D-Tic7, CpG8]des-Arg9-bradykinin | - |
Oryctolagus cuniculus | |
0.00096 | - |
L-Lys-L-Lys-[Hyp3, CpG5, D-Tic7, CpG8]des-Arg9-bradykinin | - |
Oryctolagus cuniculus | |
0.0022 | - |
D-Arg-L-Lys-[Hyp3, CpG5, D-Tic7, CpG8]des-Arg9-bradykinin | - |
Homo sapiens | |
0.00487 | - |
L-Lys-L-Lys-[Hyp3, CpG5, D-Tic7, CpG8]des-Arg9-bradykinin | - |
Homo sapiens |