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Literature summary for 3.4.11.2 extracted from

  • Tsukamoto, H.; Shibata, K.; Kajiyama, H.; Terauchi, M.; Nawa, A.; Kikkawa, F.
    Aminopeptidase N (APN)/CD13 inhibitor, Ubenimex, enhances radiation sensitivity in human cervical cancer (2008), BMC Cancer, 8, 74.
    View publication on PubMedView publication on EuropePMC

Application

Application Comment Organism
medicine inhibition of CD13 by ubenimex enhances the effectiveness of radiotherapy, with ubenimex acting as a radiosensitizer both in vitro and in vivo Homo sapiens
medicine treatment of mice with a combination of radiation and ubenimex results in significant prolongation of the tumor-doubling time Mus musculus

Inhibitors

Inhibitors Comment Organism Structure
ubenimex
-
Homo sapiens
ubenimex
-
Mus musculus

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
isoform CD13
-
Mus musculus
-
isoform CD13
-

Source Tissue

Source Tissue Comment Organism Textmining
HeLa cell
-
Homo sapiens
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
L-Ala-4-nitroanilide + H2O
-
Mus musculus L-Ala + 4-nitroaniline
-
?
L-Ala-4-nitroanilide + H2O
-
Homo sapiens L-Ala + 4-nitroaniline
-
?