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Literature summary for 3.4.11.18 extracted from

  • Lazarus, D.D.; Doyle, E.G.; Bernier, S.G.; Rogers, A.B.; Labenski, M.T.; Wakefield, J.D.; Karp, R.M.; Clark, E.J.; Lorusso, J.; Hoyt, J.G.; Thompson, C.D.; Hannig, G.; Westlin, W.F.
    An inhibitor of methionine aminopeptidase type-2, PPI-2458, ameliorates the pathophysiological disease processes of rheumatoid arthritis (2008), Inflamm. Res., 57, 18-27.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
[(1R)-1-carbamoyl-2-methyl-propyl]-carbamic acid-(3R,4S,5S,6R)-5-methoxy-4-[(2R,3R)-2-methyl-3-(3-methyl-but-2-enyl)-oxiranyl]-1-oxa-spiro[2.5]oct-6-yl ester PPI-2458, 5 mg/kg Rattus norvegicus

Organism

Organism UniProt Comment Textmining
Rattus norvegicus P38062
-
-

Source Tissue

Source Tissue Comment Organism Textmining
thymus
-
Rattus norvegicus
-

Synonyms

Synonyms Comment Organism
MetAP-2
-
Rattus norvegicus
methionine aminopeptidase type-2
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Rattus norvegicus