Cloned (Comment) | Organism |
---|---|
expression in baculoviral system | Homo sapiens |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
methyl 4-((1,2,3,4-tetrahydronaphthalene-2-carboxamido)methyl)benzoic acid | - |
Homo sapiens | |
methyl 4-([[(6-hydroxynaphthalen-2-yl)carbonyl]amino]methyl)benzoate | - |
Homo sapiens | |
methyl 4-([[(6-methoxynaphthalen-2-yl)carbonyl]amino]methyl)benzoate | - |
Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
cyano(2-methoxynaphthalen-6-yl)methyl trans-(3-phenyloxiran-2-yl)methylcarbonate + H2O | - |
Homo sapiens | ? | - |
? |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.0000018 | - |
pH 7.0, 30°C | Homo sapiens | methyl 4-([[(6-hydroxynaphthalen-2-yl)carbonyl]amino]methyl)benzoate | |
0.0000021 | - |
pH 7.0, 30°C | Homo sapiens | methyl 4-((1,2,3,4-tetrahydronaphthalene-2-carboxamido)methyl)benzoic acid | |
0.0000024 | - |
pH 7.0, 30°C | Homo sapiens | methyl 4-([[(6-methoxynaphthalen-2-yl)carbonyl]amino]methyl)benzoate |