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Literature summary for 3.2.2.22 extracted from

  • Jandhyala, D.M.; Ahluwalia, A.; Obrig, T.; Thorpe, C.M.
    ZAK: a MAP3Kinase that transduces Shiga toxin and ricin induced proinflammatory cytokine expression (2008), Cell. Microbiol., 10, 1468-1477.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
additional information 7-[3-fluoro-4-aminophenyl-(4-(2-pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-]pyrazol-3-yl))]-quinoline, i.e. DHP-2, a zipper sterile-alpha-motif kinase-specific inhibitor, blocks the SAP kinase activation induced by ricin or Shiga toxin, but is not inhibitory to the toxins Escherichia coli
additional information 7-[3-fluoro-4-aminophenyl-(4-(2-pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-]pyrazol-3-yl))]-quinoline, i.e. DHP-2, a zipper sterile-alpha-motif kinase-specific inhibitor, blocks the SAP kinase activation induced by ricin or Shiga toxin, but is not inhibitory to the toxins Ricinus communis

Organism

Organism UniProt Comment Textmining
Escherichia coli
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Ricinus communis
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