Inhibitors | Comment | Organism | Structure |
---|---|---|---|
2-formyl-17alpha-benzyl-17beta-hydroxyestra-1,3,5(10)-triene | time- and concentration-dependent inhibitor, shows more or less pseudo-first order behavior at all concentrations | Homo sapiens | |
4-fluoro-17alpha-benzyl-17beta-hydroxyestra-1,3,5(10)-triene | linear mixed-type inhibition, compound is capable of binding at sites both within and outside the active site | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
placenta | - |
Homo sapiens | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
4-methylumbelliferyl sulfate + H2O | - |
Homo sapiens | 4-methylumbelliferol + sulfate | - |
? |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.000085 | - |
2-formyl-17alpha-benzyl-17beta-hydroxyestra-1,3,5(10)-triene | pH 7.0, temperature not specified in the publication | Homo sapiens |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.00004 | - |
pH 7.0, temperature not specified in the publication | Homo sapiens | 4-fluoro-17alpha-benzyl-17beta-hydroxyestra-1,3,5(10)-triene |