Cloned (Comment) | Organism |
---|---|
- |
Homo sapiens |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
667-coumate | - |
Homo sapiens | |
KW-2581 | active site-directed irreversible steroidal inhibitor | Homo sapiens |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.00685 | - |
Estrone sulfate | 37°C | Homo sapiens | |
0.00944 | - |
dehydroepiandrosterone 3-sulfate | 37°C | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
recombinant enzyme | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
dehydroepiandrosterone 3-sulfate + H2O | - |
Homo sapiens | dehydroepiandrosterone + sulfate | - |
? | |
estrone sulfate + H2O | - |
Homo sapiens | estrone + sulfate | - |
? |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.000015 | - |
667-coumate | 37°C | Homo sapiens | |
0.000026 | - |
KW-2581 | 37°C | Homo sapiens |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.0000029 | - |
37°C | Homo sapiens | 667-coumate | |
0.000015 | - |
37°C | Homo sapiens | KW-2581 |